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8-[(2-aminopyridin-3-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(2-methoxyethyl)-9-[4-(propan-2-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
6-{3-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
2-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-8-methoxyquinoline
1-(2,4-dimethylphenoxy)-3-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-2-ol
4-[(1,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]-N,4-dimethylpentanamide
3-chloro-N-cyclopentyl-4-({1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}oxy)benzamide
2-{4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]phenoxy}propanamide
N-[1-(3-methoxyphenyl)-5-oxopyrrolidin-3-yl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
7-(3-chlorophenyl)-4-(3-fluoropropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-4-(pyridin-3-ylmethyl)piperazine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-methylfuran-3-carboxamide
1-(2-{[6-(dimethylamino)pyrazin-2-yl]oxy}hex-5-en-1-yl)piperidine-4-carboxylic acid
(2R)-2-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-phenylacetamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(oxolane-2-carbonyl)-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazine
1,1,1-trifluoro-3-{3-[3-(pyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
(1S,5R)-6-(cyclobutylmethyl)-3-[(2,5-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-dimethyl-2-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]acetamide
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]but-3-en-1-one
N,2,5-trimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-{4-[2-(2-methyl-1H-imidazol-1-yl)propanamido]phenyl}pentanamide
2-[(4-butoxyphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
2-(pyridin-2-yl)-5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]pyrimidin-4-ol
3-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-ylmethyl]-N-benzyl-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(2-methoxyacetyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
4-{[1-(ethylcarbamoyl)pyrrolidin-3-yl]methyl}benzoic acid
N-[2-(dimethylamino)ethyl]-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}furan-2-carboxamide
N-cyclohexyl-5-(1-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}ethyl)-N,4-dimethylpyrimidin-2-amine
1-[4-(benzyloxy)butyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
3-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-4-(1-ethylpiperidin-4-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
4,5-dimethyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-2-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
6-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
N-[2-(2-chloro-6-methylphenoxy)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-N-methylpyridin-2-amine
2-methyl-6-({5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}amino)heptan-2-ol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(pyridin-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(adamantan-1-yl)-1-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]ethan-1-one
N-methyl-N-propyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
(1R,9S)-5-amino-3-[4-hydroxy-3-(prop-2-en-1-yl)phenyl]-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-(4-methoxy-3,5-dimethylphenyl)-2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}acetic acid
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-dimethoxyphenyl)acetamide