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N-methyl-5-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-methyl-N-[(4-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
methyl 3-(2H-1,3-benzodioxol-4-ylmethyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-{[1-(pyrazin-2-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
5-(3-methoxyphenoxymethyl)-N-(pentan-2-yl)-1H-pyrazole-3-carboxamide
N-(1-{1-[2-(4-ethylpiperazin-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
N-[(2-chloropyridin-3-yl)methyl]-1-cyclopentyl-N-methyl-6-oxopiperidine-3-carboxamide
6-ethyl-4-[2-(2-hydroxyethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-(5-acetylthiophen-3-yl)-1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-amino-4-methyl-1,3-thiazole-5-carboxamide
2-(3-methoxypropyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidine
1-(6-hydroxy-4-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1,4-diazepan-1-yl)ethan-1-one
3,3-dimethyl-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(morpholin-4-ylmethyl)piperidin-4-ol
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
3-ethoxy-1-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]propan-1-one
N-[2-(azepan-1-yl)ethyl]-N,2-dimethyl-1-benzofuran-5-carboxamide
3-(2-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}propyl)-3,4-dihydroquinazolin-4-one
[5-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)-2-ethoxyphenyl]methanol
1'-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[3-(1H-imidazol-1-yl)propyl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
3-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)butan-1-ol
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-methanesulfonylpiperidine
4-(5-fluoro-2-methoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(5S,9aS,9bS)-5-(2-chloro-6-fluorophenyl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[3-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propan-1-one
4-{[4-(2-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-ethyl-3,5-dimethyl-1H-pyrazole
8-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane
1-(pyrimidin-2-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-amine
1-[2-(aminomethyl)morpholin-4-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
2-(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)ethan-1-ol
4-{6-[1-(pyridine-4-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
1-(2-{[(6-cyclopropylpyrimidin-4-yl)amino]methyl}morpholin-4-yl)ethan-1-one
2,6,8-trimethyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)quinoline-4-carboxamide
1-(1,4-dithiepan-6-yl)-N-phenylpiperidin-3-amine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyrrolidin-3-yl)piperidine-4-carboxamide
N,N,1-trimethyl-4-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]piperidin-4-amine
4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-1-(4-butylphenyl)-1H-pyrazole
[7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[2-methoxy-5-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
5-benzyl-3-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-methyl-N-(1-methylpiperidin-4-yl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
(1S,5S)-3-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-(1H-pyrazol-5-ylmethyl)benzamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(oxan-4-ylmethyl)amine
methyl 2-[4-(6-methoxypyrimidin-4-yl)-2-oxopiperazin-1-yl]acetate
2,6-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]quinoline-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-dihydroquinoxalin-2-one
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one