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1-(2,3-dihydro-1H-isoindol-2-yl)-2-[4-(pyrrolidine-1-sulfonyl)morpholin-3-yl]ethan-1-one
(4aS,8aR)-6-[2-(methylsulfanyl)acetyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[(5-methylpyrazin-2-yl)methyl]-9-(3-phenylpropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(2,5-dimethylbenzenesulfonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl (2S)-2-{[5-(cyclohexylcarbamoyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
4-phenyl-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-ol
2-[5-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)furan-2-yl]benzonitrile
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(9H-fluoren-2-ylmethyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-({4-hydroxy-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]azepan-4-yl}methyl)-3-methylbenzamide
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,6-dimethoxybenzamide
1-(2-oxo-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
(3S)-N,N-dimethyl-1-{[5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrrolidin-3-amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)acetamide
1-{4-[(prop-2-en-1-yl)carbamoyl]phenyl}-1H-imidazole-4-carboxylic acid
1-(3-{[(3R,4R)-1-(benzenesulfonyl)-4-hydroxypyrrolidin-3-yl]amino}propyl)pyrrolidin-2-one
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-8-fluoroquinoline
4-{1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}pyridine
3-(azepane-1-carbonyl)-5-(4-cyclopentylpiperazin-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole
2-{1-[(4-ethylphenyl)methyl]-5-(oxan-4-yl)-1H-1,2,4-triazol-3-yl}acetamide
3-{3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}pyridine
1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-4-carboxamide
N-(1-benzylpyrrolidin-3-yl)-2-ethyl-N-methylpyrimidine-5-carboxamide
2-[2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-2-carbonyl)piperidine
1-(2-methoxyphenyl)-4-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine
2-[1-(4-ethyl-5-methylthiophene-3-carbonyl)-1,4-diazepan-6-yl]acetic acid
2-(2-hydroxyethyl)-8-[(5-phenylthiophen-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-({1-[(2-chlorophenyl)methyl]piperidin-4-yl}methyl)-3-(propan-2-yl)urea
(1R,5R)-6-(5-fluoro-2-methylbenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-(4-phenyl-1,3-thiazol-2-yl)pyrrolidin-3-yl]methyl}piperidin-4-ol
2-(3,4-dichlorophenyl)-4-(3-methoxypyrazin-2-yl)morpholine
3-methyl-7-[2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(1H-1,3-benzodiazol-1-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
(3aS,6aS)-2-(5-chlorothiophene-2-carbonyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-methyl-3-{[(3-phenylprop-2-yn-1-yl)(propyl)amino]methyl}-1H-indole-2-carboxylic acid
(3S,9aR)-3-(cyclohexylmethyl)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(1H-imidazol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
2-(propylsulfanyl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3aS,6aR)-3-[2-(piperidin-1-yl)ethyl]-5-[3-(trifluoromethyl)pyridin-2-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
ethyl 1-[2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carbonyl]piperidine-2-carboxylate
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
(3S,4R)-4-(pyridin-3-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidine-3-carboxylic acid
2-cyclopentyl-8-(3-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-methoxypropanamide
ethyl 1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperidine-4-carboxylate
3-[(4-methoxyphenyl)methyl]-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine