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2-cyclopentyl-9-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
8-(2-ethoxyethyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(quinolin-8-ylmethyl)amine
2-{[3-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}carbamoyl)phenyl]amino}acetic acid
2-{2-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]-N-propylpyrimidin-2-amine
6-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
4-fluoro-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
4-[(3-fluorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
N-(2,6-dimethylphenyl)-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}benzamide
4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
1-(1,3-dihydroxypropan-2-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-(dimethylamino)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N-(1-hydroxybutan-2-yl)-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-(thiophen-2-ylmethyl)acetamide
3-fluoro-4-methoxy-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide
N-benzyl-N-butyl-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
(3aS,6aS)-2-[(2-methylpropoxy)carbonyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-chlorophenyl)-1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
5-[1-(2-cyclohexylacetyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-amino-4-{[(2S)-2,3-dihydroxypropyl]amino}quinazoline-6-carboxylic acid
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
4-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-2-methoxyphenol
N3-benzyl-1-cyclopropyl-4-oxo-N5-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]pyrazin-2-ol
N-[1-(dimethylamino)butan-2-yl]-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
1-benzyl-N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-4-carboxamide
5-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
1-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}pent-4-en-1-one
(3R,5S)-N-[3-(morpholin-4-yl)propyl]-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
methyl 2-(3-methylphenyl)-2-(1H-pyrazol-3-ylformamido)acetate
1-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
2-[(3,5-difluorophenyl)methyl]-8-(propan-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-[1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)pyrrolidin-3-yl]benzoic acid
5-(3-ethynylbenzoyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3S,4R)-1-[(3-carboxyphenyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
(2S)-2-(methoxymethyl)-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
1-acetyl-N-[2-(benzyloxy)ethyl]piperidine-3-carboxamide
1-ethyl-4-[6-phenyl-2-(pyrrolidin-1-yl)pyridine-3-carbonyl]piperazine
2-(pyridin-4-yl)-3-(pyrrolidine-1-carbonyl)pyridine
(1-{[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
4-[2-(3-methylpiperidin-1-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[3-(2-methoxybenzoyl)piperidin-1-yl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
3-benzyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenylpiperidine
N-[4-(3-fluorophenyl)phenyl]-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1-(pyridin-2-yl)ethan-1-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
(1R,5R)-6-benzyl-3-phenylmethanesulfonyl-3,6-diazabicyclo[3.2.2]nonane