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(3S,4S)-1-[3-(morpholin-4-yl)propanoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
3-methyl-7-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
[(5-ethylpyridin-2-yl)methyl](methyl)[(2-methyl-1,3-oxazol-4-yl)methyl]amine
(8R,9aS)-2-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-5-methylphenol
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
4-(4-fluorophenyl)-1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]butan-1-one
3-(2-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
N-(pyridin-2-ylmethyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
2-[3-cyclopropyl-5-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-1,2,4-triazol-1-yl]pyridine
4-(2,4-dioxoimidazolidin-1-yl)-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)benzamide
3-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}benzonitrile
[2-({4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazin-1-yl}methyl)phenyl]methanol
[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methanol
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-(2-methylphenyl)pyrrolidin-3-ol
2-(3-chlorophenyl)-N-[4-(4-{[2-(pyrazin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
{2,4,6-trimethyl-3-[(2-methyl-3-oxopiperazin-1-yl)methyl]phenyl}methyl acetate
3-methyl-6-(3-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridazine
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-[(2,3-dimethoxyphenyl)methyl]-4-{4-[2-(3-fluorophenyl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-(methoxymethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(2-hydroxypropyl)acetamide
1-{4-[4-(3-fluorophenoxy)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
1-[1'-(3-hydroxy-2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-(methoxymethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}cyclobutane-1-carboxamide
(1-{1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-4-yl}ethyl)dimethylamine
N-[(2-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-3,5-dimethyl-1H-indole-2-carboxamide
6-[(2-fluorophenyl)methoxy]-4-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
1'-(5-fluoro-1H-indole-2-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-phenyl-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}prop-2-yn-1-one
N-(4-methoxy-3-pentanamidophenyl)pyrazine-2-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-3-(4-methylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,4-oxazepan-6-ol
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2-chlorophenyl)-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-phenylpropanamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-(5-ethylthiophene-2-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(4-methyl-1,4-oxazepan-6-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N,N-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-methyl-2-(1-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)-N-[2-(oxan-2-yl)ethyl]acetamide
2,3,5,6-tetramethyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]benzamide
4-(2,2-dimethyloxane-4-carbonyl)-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{4-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1,4-diazepan-1-yl}ethan-1-one
N-[2-(4-methoxyphenyl)phenyl]-1-(6-methylpyrimidin-4-yl)piperidine-3-carboxamide