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4-[(4-methylphenyl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
N-({1-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
(1R,3S)-3-{cyclopropyl[(4-hydroxyphenyl)methyl]carbamoyl}cyclopentane-1-carboxylic acid
N-methyl-5-propyl-N-[1-(pyridin-4-yl)ethyl]thiophene-3-carboxamide
1-({[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]amino}methyl)cyclohexan-1-ol
3-(4-chlorobenzoyl)-1-(cyclohex-1-ene-1-carbonyl)piperidine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(6-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[4-phenyl-1-(pyrimidin-4-ylmethyl)-1H-imidazol-5-yl]benzoic acid
(4aS,7aR)-N-(2,5-dimethylphenyl)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-[4-(3-fluorophenoxy)piperidine-1-carbonyl]benzonitrile
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}butan-1-one
3-{1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
5-chloro-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-3-phenyl-1H-indole-2-carboxamide
2-({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)pyrimidine
2-(2-chlorophenyl)-3-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-cyclopentanecarbonyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]piperidine-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-(quinolin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-4-amino-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrrolidine-2-carboxamide
N-ethyl-2-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}acetamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)(4,4,4-trifluorobutyl)amine
3-{[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}benzonitrile
9-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(2-ethoxyphenyl)methyl]-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
1-(morpholin-4-yl)-2-[3-(4H-1,2,4-triazol-4-yl)phenoxy]ethan-1-one
7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-4-(pyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,2R,4R)-N-[3-(1H-indazol-1-yl)propyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-(3-methoxy-2,2-dimethylpropyl)cyclohex-3-ene-1-carboxamide
1-[3-(1H-pyrazol-4-yl)benzoyl]pyrrolidin-3-ol
N-(4-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)benzenesulfonamide
N3-{[4-(2-methoxyethoxy)phenyl]methyl}-N1,N1-dimethylpiperidine-1,3-dicarboxamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-(3-methylbenzoyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
ethyl 1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
1-[6-(1-hydroxyethyl)pyridin-2-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]phenyl}butan-1-ol
ethyl[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
N-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-N-methylthian-4-amine
4-(5-chloro-2-hydroxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
2-[2-(1H-imidazol-1-yl)ethyl]-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
7-(cyclobutylmethyl)-2-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
2-[3-({[1-(furan-2-ylmethyl)piperidin-4-yl]carbamoyl}amino)phenyl]-N-methylacetamide
N5-benzyl-N6-[2-(dimethylamino)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[(4-chlorophenyl)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
(3aR,6aR)-2-[(5-chlorofuran-2-yl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[3-(4-methylbenzenesulfonamido)propyl]carbamoyl}-1H-imidazole-4-carboxylic acid
1-(2-chlorobenzoyl)-4-(1-methyl-1H-1,2,4-triazol-5-yl)piperidine
[(5-ethylpyridin-2-yl)methyl]({[3-(3-fluorophenyl)oxolan-3-yl]methyl})amine
[(3R,4S)-1-[(3-chloro-4-ethoxyphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol