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6-(2-chlorophenyl)-2-(3-{[(3R)-3-hydroxypiperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(2S,4S)-4-amino-N-ethyl-1-(4-methoxy-2-methylbenzoyl)pyrrolidine-2-carboxamide
4-{6-[4-(pyridin-2-ylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-(thiophen-3-ylmethyl)piperidine
N,1-bis(propan-2-yl)-2-(quinolin-6-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
3-[(dimethylamino)methyl]-1-{[4-(2-phenylethoxy)phenyl]methyl}piperidin-3-ol
{2-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]phenyl}methanol
1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
N-[(2-aminopyridin-3-yl)methyl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-propyl-3-(pyrrolidine-1-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3R,4S)-1-[2-(morpholin-4-yl)-2-oxoethyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[(1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]pyridine
4-cyclobutyl-2-(3-ethylpiperazin-1-yl)-6-methylpyrimidine
5-fluoro-N4,N4-dimethyl-N2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidine-2,4-diamine
5-(2-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-{[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzothiazol-2-one
N-[(5-methylpyrazin-2-yl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethoxy]benzamide
3-hexyl-8-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,4S)-4-(5-methylfuran-2-yl)-1-(oxan-4-yl)pyrrolidin-3-amine
1-{7-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
4-chloro-2-({[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amino}methyl)phenol
4-ethyl-1-methyl-3-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-methyl-2-(4-methyl-1,4-diazepan-1-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
4-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1-methylimidazolidin-2-one
({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amine
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
1-(3-hydroxy-4-methylbenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
1-cyclohexyl-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(4-propylphenyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-cyclopentyl-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
6-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-{2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
4-(2,3-dihydro-1-benzofuran-7-carbonyl)-1-methylpiperazine-2-carboxylic acid
4-[(3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,2-oxazol-5-yl)methyl]morpholine
2-{4-[(8-methoxy-2H-chromen-3-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
3-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-5-(2-methylphenyl)-1,2,4-triazine
5-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
2-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(1-phenylethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
ethyl 1-[(2-hydroxyphenyl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
2-{3-tert-butyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3,5,6-trimethylpyrazine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(2-methoxyphenoxy)azetidine
1-cyclopropanecarbonyl-3-[2-(3-fluorophenyl)ethyl]piperidine
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
3-(5-fluoro-2-methoxybenzoyl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
N-(3-methoxyphenyl)-3-[1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-4-yl]propanamide
7-{2-methyl-2-[5-methyl-2-(propan-2-yl)phenoxy]propanoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one