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2-(propan-2-yl)-1-[2-(pyrrolidin-1-yl)benzoyl]-2,5-dihydro-1H-pyrrole
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methyl-7-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2,8-dimethyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)cyclopropanamine
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-[(2-fluorophenyl)methyl]piperazin-2-one
1-[2-(2-chloro-4-fluorophenyl)acetyl]-4-propyl-1,4-diazepan-5-one
2-{1-[1-(cyclopropanesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
1-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)piperidine-3-carboxamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(trifluoromethyl)benzamide
2,2-diphenyl-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2-(pyridin-3-yl)acetamide
2-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
methyl(oxan-4-ylmethyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[3-(methylsulfanyl)phenyl]-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
N-(2-hydroxyethyl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
4-(2-methyl-5-propylpyrimidin-4-yl)piperazine-2-carboxylic acid
1-cyclobutyl-N-(4-fluorophenyl)piperidin-3-amine
(4aS,7aR)-1-(2-ethoxyacetyl)-4-(3-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyridine-2-carbonitrile
1-[({2-[(2-chlorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)amino]propan-2-ol
propan-2-yl N-{[(3S,4S)-3-hydroxy-1-(1-hydroxycyclopentanecarbonyl)piperidin-4-yl]methyl}carbamate
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-3-[2-(1H-imidazol-4-yl)ethyl]urea
2-[3-({cyclopropyl[(3-ethoxyphenyl)methyl]amino}methyl)-1H-indol-1-yl]acetamide
2-[1-(3-fluoro-2-methoxybenzoyl)pyrrolidin-3-yl]benzoic acid
N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
[(3-chlorophenyl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
2-{2-[(3-fluorophenyl)methoxy]phenyl}-N-methylpyridine-3-carboxamide
(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(3-hydroxypyridine-2-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
(3R,4S)-4-cyclopropyl-1-[6-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
N-[(4-fluorophenyl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-4H-chromen-4-one
(2R)-2-acetamido-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}butanamide
(4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholin-2-yl)methanamine
(1R,5S,6R)-3-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-N-(1H-imidazol-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propan-2-ol
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,4-dioxane-2-carboxamide
N-cyclopentyl-5-[(3-methoxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(2-hydroxyethyl)-2-(7-methoxy-4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{3-cyclopentyl-5-[4-(2,4-dioxoimidazolidin-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-(2-fluoroethyl)-3-{[1-(4-hydroxyphenyl)ethyl]sulfamoyl}benzamide
1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methylpiperidine-3-carboxamide
1-(methoxymethyl)-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-phenylpyrrolidin-3-yl]cyclobutane-1-carboxamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(quinolin-4-ylmethyl)propanamide