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1-[3-(diethylamino)pyrrolidin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
1-methyl-2-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
2-cyclopropyl-5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]pyrimidine
3-[(3-chlorophenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(pyridin-2-ylsulfanyl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-butyl-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
[1-(5-methyl-4-{methyl[2-(4-methylphenoxy)ethyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperidin-2-yl]methanol
4-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-oxopiperazin-1-yl}benzonitrile
(3R)-1-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}pyrrolidin-3-ol
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]cyclobutanecarboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(5-methyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
2-(5-amino-4H-1,2,4-triazol-3-yl)-N-[(4-methoxynaphthalen-1-yl)methyl]-N-methylacetamide
4-chloro-N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-methyl-1H-pyrazole-5-carboxamide
4-(4-{[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
N-{[4-(dimethylamino)oxan-4-yl]methyl}-4-methylpyrimidin-2-amine
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)-N-propylpiperidine-3-carboxamide
{4-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}methanol
2-[2-(4-methylpentyl)morpholine-4-carbonyl]benzene-1,3-diol
1-[2,2-dimethyl-1-(3-methylthiophen-2-yl)cyclopropanecarbonyl]-4-hydroxypiperidine-4-carboxylic acid
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(cyclopropanesulfonyl)piperidine
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-3-(4-methylphenyl)propanamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-{[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
N-methyl-3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
4-(benzyloxy)-1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperidine
5-(4-chlorophenyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-1,2,4-triazin-3-amine
2-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-5-methylpyrazine
5-chloro-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-(dimethylamino)-8-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
[(3R,4S)-1-{[3-(2-methylphenyl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-ethyl-5-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidin-2-amine
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-4-(methoxymethyl)piperidine
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(3-fluorophenyl)ethyl]amine
4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-2-methoxyphenol
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(propylcarbamoyl)piperidine-3-carboxylate
3-[3-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)propyl]pyridine
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
N-(5-methyl-1,3-thiazol-2-yl)-5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
4-{[6-(2-ethoxypyridin-3-yl)pyridin-3-yl]methyl}morpholine
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-3-(pyridin-4-yl)propanamide
4-[5-(2-methoxy-3,5-dimethylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]-1-methylpiperidine
(1S,5R)-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}[1-(2-methoxyphenyl)ethyl]methylamine