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2-(6-methoxynaphthalen-2-yl)-4-(1,3-thiazol-2-yl)morpholine
2-[methyl(pyridin-3-ylmethyl)amino]-N-[(1-phenylcyclopentyl)methyl]acetamide
3-(1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}azetidin-3-yl)pyridine
1-cyclobutyl-3-[4-(trifluoromethyl)benzoyl]piperidine
2-butyl-8-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(4-fluorophenyl)methyl]-1-[3-(1H-imidazol-1-yl)propyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[1-ethyl-2-(2-fluorophenyl)-7-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
2-(2,3-dimethoxyphenyl)-2-[4-(pyridin-2-yl)piperazin-1-yl]acetic acid
1-[(2,6-difluorophenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
(1S,5R)-6-benzyl-3-[2-(pyridin-2-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(4aS,8aR)-1-(2-aminoethyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-3-carboxamide
(5S,9aS,9bS)-5-(1-ethyl-1H-pyrazol-4-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(4-ethylpiperazin-1-yl)-N-[3-(propan-2-yloxy)propyl]-2,3-dihydro-1H-indene-2-carboxamide
N-cyclohexyl-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
8-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(2S,4R)-4-(dimethylamino)-1-[(4-ethylphenyl)methyl]pyrrolidin-2-yl]methanol
3-[(3-hydroxy-3-phenylpyrrolidin-1-yl)methyl]-6-methyl-1,2-dihydroquinolin-2-one
methyl 3-[propyl(pyridin-3-ylmethyl)carbamoyl]benzoate
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrimidin-2-amine
6-methyl-3-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-[8-(1H-indol-2-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
9-(3,5-dimethylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(1-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}azetidin-3-yl)morpholine
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]benzoic acid
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
2-(dimethylamino)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(2-methylphenyl)acetamide
3-hydroxy-S-(2-pentanoyl-1,2,3,4-tetrahydroisoquinolin-7-yl)butane-1-sulfonamido
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-[4-(morpholin-4-yl)piperidin-1-yl]propan-1-one
5-ethyl-N-[(1S)-1-(3-methoxyphenyl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-methoxy-9-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecane
3-{1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-(2-methylpropyl)-1H-pyrazole
(2S)-2-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-hydroxypropan-1-one
5-(2,6-difluorophenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-cyclobutyl-6-(4-fluorophenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-[(2-chloro-6-fluorophenyl)methyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(cyclopentyloxy)phenyl]methyl}pyrrolidin-3-amine
methyl 3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetamido]methyl}-5-[(2E)-3-phenylprop-2-enamido]benzoate
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
5-[2-(4-phenylpiperidin-1-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
9-{2-[ethyl(methyl)amino]acetyl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[2-(4-methyl-1H-imidazol-2-yl)ethyl]({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
3-[(4-fluorophenyl)methyl]-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylic acid
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
2-amino-3-ethyl-N-[3-(pyridin-2-yl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N3-benzyl-1-cyclopropyl-N5-[(4-fluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3R,9aR)-3-benzyl-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(6-methylpyridine-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol