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3-(4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)pyridine
(2R,4S)-4-hydroxy-1-[(3,4,5-trimethoxyphenyl)methyl]piperidine-2-carboxylic acid
(3S,4R)-1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(4-methylphenyl)-N-{2-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
methyl 2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(5-methoxyfuran-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
N-[(2R,3R)-1'-(1-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(1,2-oxazinan-2-yl)propan-1-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[3-(methoxymethyl)pyrrolidin-1-yl]propan-1-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-[3-(2-methylpropyl)pyrrolidin-1-yl]pyridine-2-carboxamide
N-[5-(oxolan-2-yl)-1,3,4-thiadiazol-2-yl]-2-{[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]amino}acetamide
2,5-dimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
(3S,4S)-4-cyclopropyl-1-(2-methylpyridin-4-yl)pyrrolidine-3-carboxylic acid
(1S,5R)-3-benzoyl-6-(5-propyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-hydroxy-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
3-(1-{1-[(2R)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
8-(4-aminopyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-9-(1H-1,2,4-triazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-phenoxyethan-1-one
N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}ethan-1-one
9-methoxy-N-[(2-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-2-(thiophen-2-ylmethyl)propan-1-ol
(3S,4R)-3-ethyl-4-methyl-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-ol
3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N-methylpropanamide
4-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(4-fluorophenyl)-1H-pyrazole
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-N-(1-benzylpyrrolidin-3-yl)propanamide
(3S)-1-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-ethylbenzamide
(3S,9aR)-3-benzyl-2-methyl-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(3,4-dimethylphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
N-({1-[(2-phenylethyl)carbamoyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
1-[(2-methylphenyl)methyl]-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-(pentan-2-yl)-8-[2-(1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(cyclohexylmethyl)-N3-(2,2-dimethyloxan-4-yl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-{2-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(2-ethyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazole
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-3-(morpholin-4-yl)propan-1-one
1-[1-(2,3-difluoro-4-methylbenzoyl)piperidin-3-yl]-2-phenylethan-1-one
(1S,5R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(pyridin-3-yl)acetamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
N-[(4-chlorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-({4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)piperidin-3-amine
4-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-methylpiperidin-4-ol
(3S)-3-ethyl-4-(2-phenylmethanesulfonylbenzoyl)morpholine