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3-[3-(3-oxopiperazin-1-yl)propyl]-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
(3aS,6aR)-5-[(2-ethylphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N2-[2-(3-methylthiophen-2-yl)ethyl]pyrrolidine-1,2-dicarboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]-1H-pyrazole-3-carboxamide
N-[(2R)-1-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1-oxopropan-2-yl]acetamide
4-[2-(piperidine-1-carbonyl)phenoxy]-1-(thiolan-3-yl)piperidine
6-methyl-3-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-2-ol
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-(morpholin-4-yl)butan-1-one
4-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-1-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[2-(oxolan-3-yl)ethyl]piperidine
N-[1-(methoxymethyl)cyclopentyl]-3-(1,2-oxazinan-2-yl)propanamide
N-[(3S,4R)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-propylpyrrolidin-3-yl]acetamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
2-{2-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
(4S)-3,3,4-trimethyl-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-ol
1-{2-[4-(2,2-diphenylethyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
2-amino-6-(2-methylbutan-2-yl)-4-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]pyridine-3-carbonitrile
2-methoxy-4-({4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenol
1-methoxy-8-[(3-phenoxyphenyl)methyl]-1,8-diazaspiro[4.5]decan-2-one
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]quinoxaline
4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoropyrimidin-4-yl]morpholine
N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-2-(methylsulfanyl)propanamide
1'-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
(2S,4R)-4-(dimethylamino)-1-{[4-(methylsulfamoyl)phenyl]methyl}pyrrolidine-2-carboxylic acid
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methylbutanamide
N-{2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}pyridin-3-amine
1-[4-(1H-indol-2-yl)phenyl]-N-(oxan-4-yl)piperidin-4-amine
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amine
N-(2H-1,3-benzodioxol-5-yl)thiomorpholine-4-carboxamide
1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]propanoic acid
(3R,5R)-5-(pyrrolidine-1-carbonyl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)piperidine-3-carboxamide
4-(dimethylamino)-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-[6-(3-methoxypiperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]azepane
1'-(1,3-benzothiazole-6-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(cyclopropylmethyl)-1-(2-methyl-5-propylpyrimidin-4-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
6-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
8-(1-methyl-1H-pyrazole-4-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-ethyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
3-{[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(methyl)(propan-2-yl)amine
3-amino-1-[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]pyrrolidine-3-carboxylic acid
2-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1H-indole
(1R,9S)-5-amino-3-(3-fluoro-2-methylphenyl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile