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(2S)-N-methyl-N-(quinolin-4-ylmethyl)piperidine-2-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(2-methyl-1H-indol-1-yl)propanamide
3-{4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-ethyl-3-{2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
3-(4-benzyl-1H-pyrazol-5-yl)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidine
2-[(3-fluorophenyl)methyl]-4-[4-(2,3,4-trimethoxybenzoyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-benzyl-3-{1-[2-(1H-imidazol-1-yl)acetyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-methylpropyl)-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]amino}propan-1-ol
5-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
3-[2-(dimethylamino)-2-(4-methylphenyl)acetamido]propanoic acid
(3R,4R)-3,4-dimethyl-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]pyrrolidin-3-ol
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-methylfuran-2-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidine-3-carboxamide
4-(2-methoxyethyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine
(9aR)-8-[(3-fluoro-4-methylphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-cyclopropyl-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-1-[(4-fluorophenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
3-(azepane-1-carbonyl)-5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-1,4-dihydropyridin-4-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-propylpyrrolidin-3-yl]-4-ethyl-5-methylthiophene-3-carboxamide
3-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}benzonitrile
[(1S,3S,3aS,6aR)-3-[4-(1H-imidazol-1-yl)phenyl]-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
(2S,4R)-4-amino-N-ethyl-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidine-2-carboxamide
N-[(4-methoxyphenyl)methyl]-4-oxo-N-propyladamantane-1-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
(2S,4S)-N-methyl-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(6-methylpyridin-2-yl)methyl]benzamide
3-[4-(3-chlorophenyl)piperazine-1-carbonyl]-2-cyclopropyl-1-[(2-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-3-(4-methylpiperidine-1-carbonyl)-1,4-dihydropyridin-4-one
4-(4-fluorophenyl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-ol
N-{2-[4-(furan-3-ylmethyl)morpholin-2-yl]ethyl}-3-hydroxy-2-methylbenzamide
N'-cyclohexyl-N'-methyl-N-[(1-methylpiperidin-4-yl)methyl]butanediamide
N-ethyl-N-methyl-3,3-diphenylpiperidine-1-sulfonamide
4-[cyclopropyl(4-methylpyridin-2-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
(1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
1-(4-methoxybenzoyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
4-[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-4-phenylpiperidine
N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-[(3-methoxyphenyl)methyl]-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decane
N,N-diethyl-5-(4-phenyl-1H-imidazol-1-yl)furan-2-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2,2,2-trifluoroethyl)piperidine-4-carboxamide
2-methoxy-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N-cyclohexyl-N-(2-hydroxyethyl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
8-[2-(2-chloro-6-fluorophenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2,2-dimethylpropan-1-one