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N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrrolidine-1-sulfonamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide
2-[(4-methoxyphenyl)methyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,3-benzoxazole-6-carboxamide
1-methyl-8-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[1-(1-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
N-cyclopropyl-1-[1-(3-methylbutyl)piperidin-4-yl]piperidine-3-carboxamide
2-cyclopropyl-3-oxo-N-[4-(propan-2-yl)phenyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-5-methoxyphenol
3-methyl-N-(1-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
(1S,5R)-6-(4-fluoro-2-methylbenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-ethylacetamide
8-cyclopropanecarbonyl-2-(4-fluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(azocane-1-carbonyl)-N-[(3R)-pyrrolidin-3-yl]benzene-1-sulfonamide
2-methyl-4-propyl-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
N-[1-(3-methylphenyl)piperidin-4-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(4-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
5-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-2-(3-methylphenyl)pyrimidine
2-[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[(2-methoxyphenyl)methyl]acetamide
(1S,5R)-3-(3-hydroxypyridine-2-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}morpholine
8-[2-(methylamino)pyridine-3-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
7-(6-chloroquinolin-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
3-butyl-1-methyl-4-[2-(pyrrolidin-1-yl)benzoyl]piperazin-2-one
2-(3-chlorophenyl)-2-hydroxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
5-{[4-(furan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazole
6-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-[2-(1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
3-{ethyl[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]amino}-1λ6-thiolane-1,1-dione
(3S,4S)-1-[2-(benzylsulfanyl)-4-hydroxypyrimidine-5-carbonyl]-4-methylpiperidine-3,4-diol
methyl 3-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2,4-dimethylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(4-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-ethyl-1-methyl-3-[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-[3-({[(2-chloro-6-fluorophenyl)methyl]amino}methyl)-5-(piperidine-1-carbonyl)phenyl]methanesulfonamide
1-methyl-4-({1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)piperazine
N-(3,4-dimethylphenyl)-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-3-amine
2-(dimethylamino)-1-[4-(3-hydroxyphenyl)piperazin-1-yl]-2-(4-methylphenyl)ethan-1-one
1-(4-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
1-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazole-5-carbonyl]-1,2,3,4-tetrahydroquinoline
4-[1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
N,N,4-trimethyl-2-[5-(pyrrolidin-2-yl)thiophene-2-amido]-1,3-thiazole-5-carboxamide
methyl 7-oxo-3-(oxolane-2-carbonyl)-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[4-(4-acetylphenyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
1-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
1-{2-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one