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N-(3-cyclopentylpropyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
methyl 1-({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperidine-4-carboxylate
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
4-[(3-methoxyphenyl)methyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-chlorobenzoyl)-N-(2-phenylethyl)piperidine-1-carboxamide
1-[3-(2-methoxyphenyl)propanoyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
N,N,4-trimethyl-3-({[2-(pyridin-2-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(3-fluorophenyl)-3-{1-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{3-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
N-[(3R,4S)-4-cyclopropyl-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amine
2-[(1S,5R)-3-(3-cyano-2-methoxypyridin-4-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N3-(butan-2-yl)-1-cyclopentyl-4-oxo-N5-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(3,4-difluorophenyl)-5-(2,3-dihydro-1-benzofuran-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
ethyl 1-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-[(5-ethylpyridin-2-yl)methyl]-4-hydroxy-N-methyl-2-(phenoxymethyl)pyrimidine-5-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-(3-hydroxypropyl)-N-methyl-1,2-oxazole-3-carboxamide
3-benzyl-5-{imidazo[2,1-b][1,3]thiazol-6-yl}-1H-1,2,4-triazole
2-(4-fluorophenyl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[4-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[2-(4-methoxyphenyl)ethyl]-N-[(5-methylfuran-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-(3-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[1-(thiophen-3-ylmethyl)piperidin-3-yl]methyl}furan-2-carboxamide
[2-(2-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenoxy)ethyl]dimethylamine
ethyl 2-[1-benzyl-4-(4-fluorobenzenesulfonyl)piperidin-4-yl]acetate
4-({2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}methyl)-3-methylpiperazin-2-one
methyl({[5-(oxan-2-yl)furan-2-yl]methyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-{[(6-methylpyridin-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
2-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyridin-3-ol
8-[4-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S,4S)-1-[(2-fluorophenyl)methyl]-4-propanamidopyrrolidine-2-carboxylate
1-(cyclohexylmethyl)-N-cyclopropyl-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(2-methoxyethyl)-6-[3-(pyridine-3-carbonyl)piperidine-1-carbonyl]-1,3-benzoxazole
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-(4-fluorophenyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
4-[(2,4-difluoro-3-methoxyphenyl)methyl]-3-ethylmorpholine
6-fluoro-4-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-1,2-dihydroquinolin-2-one
1-(3-phenylpropyl)-4-(pyrrolidin-3-yl)piperazine
N-{1-[1-(2-cyclohexylacetyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylthiophene-3-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{2-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]phenoxy}ethan-1-ol
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-(morpholin-4-yl)pyridine-3-carboxamide
[(3S,5R)-1-(3,6-dimethylpyrazin-2-yl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
(4aS,7aR)-1-(6-hydroxyhexyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-(1H-indol-1-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
1-(cyclohexylmethyl)-N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-6-oxopiperidine-3-carboxamide
(2R,3R,6R)-5-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(cyclopropylmethyl)-1-[(2-methylphenyl)methyl]-N-propyl-1H-1,2,3-triazole-4-carboxamide