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1-(4-ethylpiperazin-1-yl)-3-[3-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-1,2,3-triazole
N-[1-(2-ethyl-1H-imidazol-1-yl)propan-2-yl]-1-(4-methylbenzoyl)piperidin-4-amine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}oxane-4-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
2-{[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
(2-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-2-yl}ethyl)dimethylamine
(3R,4S)-1-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(propan-2-yl)pyrrolidin-3-amine
3-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]propanoic acid
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-(morpholin-4-yl)ethan-1-one
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethylpropanamide
13-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
9-[2-(2-methoxyethoxy)acetyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
(3aS,6aS)-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
1-methyl-2-phenyl-4-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazine
4-ethyl-3-(piperidin-3-yl)-1-{[4-(propan-2-yl)phenyl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
methyl 2-({3-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]phenyl}amino)acetate
1-(4-fluoro-2-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenyl)ethan-1-one
(3S,9aR)-8-(4-chlorobenzenesulfonyl)-3-(cyclohexylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 3-({2-[(4-methoxyphenyl)methyl]-1,3-benzoxazol-6-yl}formamido)propanoate
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethyl-4-oxobutanamide
3-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-N-(2,3-dimethylphenyl)-3-oxopropanamide
4-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-N-(pyridin-3-yl)benzamide
N-(2-methoxyethyl)-4-{[2-(4-methoxyphenyl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
N5-(2,3-dihydro-1H-inden-2-yl)-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-methyl-4-{3-methyl-5-[5-(pyrrolidin-2-yl)thiophen-2-yl]-1H-1,2,4-triazol-1-yl}pyridine
2-{1-[(4-methylphenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-yl}ethan-1-ol
N-[3-(3-chlorophenyl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
3-benzyl-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one
5-[5-(1-cyclohexyl-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
2-(4-methoxyphenoxymethyl)-N-(1-phenylethyl)-1,3-oxazole-4-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-(pyridin-2-yl)acetamide
6-{4-[(dimethylamino)methyl]phenoxy}-N-ethyl-N-methylpyridine-3-carboxamide
(1R,5R)-3-methanesulfonyl-6-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
4-(2,3-dihydro-1H-inden-2-yl)-N-(4-fluoro-3-methoxyphenyl)piperazine-1-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
5-(1-cyclopentylpyrrolidin-2-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}thiophene-2-carboxamide
4-({[(3-hydroxypiperidin-3-yl)methyl]carbamoyl}amino)-N-(2-methoxyethyl)-3-methylbenzamide
3-methyl-1-(2-methylpropyl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazin-2-one
3-[(3,6-dimethyl-1-benzofuran-2-yl)formamido]-N-(2-methoxyphenyl)propanamide
2-(4-benzyl-1-cyclohexylpiperazin-2-yl)ethan-1-ol
4-benzyl-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,8aS)-1-[(4-methoxyphenyl)methyl]-6-[3-(2-oxoimidazolidin-1-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
8-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione