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2-(2,3-dimethoxyphenyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
4-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-amine
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(3-methoxyphenyl)ethyl]propanamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-(1,3-thiazol-2-ylmethyl)piperidin-4-amine
2-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}-4,6-dimethylpyrimidine
2-(6-methoxypyridin-3-yl)-5-propylpyrimidine
N-[(5-fluoro-1H-indol-2-yl)methyl]-1-(furan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
5-[2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetyl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
1-[4-(4-methylpyridin-2-yl)piperazin-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
(3aR,5S,6S,7aS)-2-(1H-1,3-benzodiazol-2-ylmethyl)-octahydro-1H-isoindole-5,6-diol
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2-(thiophen-2-yl)-1,3-thiazole
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
[(2-butoxy-3-methoxyphenyl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
5-ethyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
2-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-6-fluoro-1H-1,3-benzodiazole
1-(1H-indazol-6-yl)-3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
5-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-N,N-dimethylpyrimidin-2-amine
4-chloro-3,5-dimethyl-1-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-pyrazole
2-[(4-chlorophenyl)methyl]-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
N-(2,3-dihydro-1H-inden-5-yl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
1-(1,3-benzothiazole-6-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-{2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-oxoethyl}pyrrolidin-2-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
5-chloro-3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
(3S,4R)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
[(5-fluoro-1H-indol-2-yl)methyl](methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
7-[(4-fluorophenyl)methyl]-2-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-({1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
2-(4-acetylpiperazin-1-yl)-2-(2-ethoxyphenyl)acetic acid
N-methyl-N-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}methanesulfonamide
butyl 2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxylate
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]acetic acid
N-[2-(azepan-1-yl)ethyl]-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(2,3-difluorophenyl)ethan-1-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine
3-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-4,5,6-trimethyl-1,2-dihydropyridin-2-one
4-(2H-1,3-benzodioxol-5-yloxy)-1-(4-methylpyridin-2-yl)piperidine-4-carboxylic acid
1-[(4-phenylphenyl)methyl]-3-(1H-pyrazol-5-yl)piperidine
6-(1H-indole-2-carbonyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(5-{1-[cyclohexyl(methyl)amino]ethyl}-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
(2S)-2-{[(5-fluoro-2-methoxyphenyl)carbamoyl]amino}-3-methylbutanamide
4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-[(4-methylphenyl)methyl]-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
ethyl 4-[5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-amido]piperidine-1-carboxylate