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3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(3-methylbutyl)carbamoyl]pyrrolidine-2-carboxylic acid
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(propan-2-yl)pyridazine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]methanol
3-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
7,8-dimethyl-3-[1-(3-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-(4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)imidazolidine-2,4-dione
N-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,5-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-hydroxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)propanamide
1-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-4-(2-methylphenyl)piperazine
N-cyclopropyl-4-methoxy-3-{[1-(1,3-thiazol-2-yl)piperidin-4-yl]oxy}benzamide
methyl 6-benzyl-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1R,9aR)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
2-[2-(dimethylamino)ethyl]-9-[2-(3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(4-methoxy-2-methylphenyl)-3-(3-methylthiophene-2-carbonyl)piperidine-1-carboxamide
dimethyl(2-{4-[2-(trifluoromethyl)benzoyl]morpholin-2-yl}ethyl)amine
N-{1-[1-(pyridin-2-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]propyl}furan-2-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(2S)-3-{[7-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}propane-1,2-diol
2-{1-[(3,5-dimethylphenyl)methyl]azetidin-3-yl}pyridine
6-{3-oxo-3-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propyl}-2,3,4,5-tetrahydropyridazin-3-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
1-ethyl-3-(2-methylpropyl)-N-(2-oxoazepan-3-yl)-1H-pyrazole-5-carboxamide
2-(2-methylpyrrolidin-1-yl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridine
2-(3-phenylpropyl)-8-(thiophene-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazole
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-(morpholin-4-yl)-N-(oxolan-2-ylmethyl)benzamide
3-[(dimethylamino)methyl]-1-[(1-ethyl-1H-indol-6-yl)methyl]piperidin-3-ol
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
2-(2-chloro-6-fluorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-4-(1H-imidazol-1-yl)benzamide
5-butyl-4-[2-(1H-imidazol-1-yl)acetyl]-1-(2-methoxyphenyl)piperazin-2-one
3-methyl-N-(1-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
7-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
N-({1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
1-{2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-phenylpyrrolidin-3-ol
(3aR,6aR)-2-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-fluorophenyl)-2-{[(naphthalen-1-ylmethyl)amino]methyl}phenol
(3S,4S)-1-(3-cyano-2-methoxypyridin-4-yl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
3-(4-chlorophenyl)-2-({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-1-ol
(2S)-2-amino-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(1,3-thiazol-4-yl)propanamide
N3-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidine-1,3-dicarboxamide
4-[2-(3-hydroxyphenyl)acetyl]-1-(2-methylphenyl)piperazin-2-one
7-(3,6-dimethylpyrazin-2-yl)-4-(2-hydroxypyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol