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2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
3-[5-(2-methoxy-6-methylphenyl)-1,2,4-oxadiazol-3-yl]pyridazine
N,N-dimethyl-2-(1-{3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-pyrazol-4-yl)quinoline-4-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-(quinolin-2-ylmethyl)piperidine-4-carboxamide
2-(dimethylamino)-N-[1-(1H-indol-2-yl)ethyl]-N,4-dimethylpyrimidine-5-carboxamide
methyl 1-methoxy-8-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N,4-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,3-thiazole-5-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1,3-benzothiazole-5-carboxamide
1-{4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)azetidin-3-ol
1-(3,5-difluorophenyl)-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(4aS,7aR)-1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(azepan-1-yl)ethyl]-6-oxo-N-(propan-2-yl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[3-(2,3-dihydro-1H-indol-1-yl)propyl]amine
N-({3-[(1E)-3,3-dimethylbut-1-en-1-yl]phenyl}methyl)propanamide
2-{[(2-chloro-5-methylphenyl)carbamoyl]amino}-N,N,3-trimethylbutanamide
N-(1-methyl-5-oxopyrrolidin-3-yl)-2,2-diphenylacetamide
5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-2-[4-(methylsulfanyl)phenyl]-1,3-oxazole
3-hydroxy-3-{[methyl(thiophen-3-ylmethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
3-(2-fluorophenyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-phenylpropanamide
N-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}-1-methanesulfonylpiperidin-4-amine
1-(2-methylphenyl)-4-(oxane-4-carbonyl)-1,4-diazepane
2-(benzyloxy)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,3-thiazole-5-carboxamide
4-[2-(azocan-1-yl)acetyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-(3-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
1-{1-[(2-ethylphenyl)methyl]piperidin-4-yl}pyrrolidin-2-one
2-({[(3R,4R)-1-(2,3-difluoro-4-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(5-methoxyfuran-2-carbonyl)piperidine
(1R,3S)-3-[3-(2-methoxyethyl)-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl]cyclopentan-1-amine
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
N-[1-(diethylcarbamoyl)azepan-3-yl]-1,3-benzothiazole-6-carboxamide
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
5-(6-methoxypyridin-3-yl)-2-methyl-1,3-benzothiazole
(2S,4S)-4-acetamido-N,N-diethyl-1-[(3-fluoro-4-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
N'-(2-fluoro-5-methylphenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}butanediamide
4-(4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)piperidin-4-ol
N-(3-chloro-4-propanamidophenyl)pyridazine-4-carboxamide
(2R,6S)-4-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
N-{2-chloro-4-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]phenyl}-2-methoxyacetamide
2-methyl-N-(4-{methyl[1-(1,3-thiazol-2-yl)ethyl]carbamoyl}phenyl)furan-3-carboxamide
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
1-(4-methylquinazolin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-4-carboxamide
3-(1H-1,2,3-benzotriazol-5-yl)-1-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)urea
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-2-(2-oxoazepan-1-yl)acetamide
{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
2-(4-methylphenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}quinoline
ethyl 1-(4-ethenylbenzoyl)-4-(2-phenylethyl)piperidine-4-carboxylate