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N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N,N-bis(2-methylpropyl)acetamide
2-cyclopropyl-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)pyrimidine-5-carboxamide
N-{[1-(1H-indol-3-ylmethyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(4-methyl-1,3-thiazol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-(1-{3-[(2,6-dichlorophenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}ethyl)pyrrolidin-2-one
1-(3-methyl-1H-pyrazole-4-carbonyl)-4-(4-methylbenzenesulfonyl)piperazine
3-fluoro-2-(2-fluoro-3-methoxyphenyl)pyridine
1-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}azetidin-3-yl)-2-methylpiperidine
3-cyano-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzene-1-sulfonamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
4-oxo-5-phenoxy-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,4-dihydropyridine-3-carboxylic acid
5-{2-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(azepan-1-yl)-2-phenylethyl]quinoxaline-6-carboxamide
N-(3-methoxypropyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-[(diethylamino)methyl]-N-(2-hydroxyethyl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
5-(3-methoxyphenoxymethyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-pyrazole-3-carboxamide
3-({2-[(4-fluorophenyl)methyl]morpholin-4-yl}methyl)-N-methyl-1,2,4-oxadiazole-5-carboxamide
3-[(3R,4S)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(2R)-2-amino-N-(isoquinolin-5-ylmethyl)-N,4-dimethylpentanamide
3-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
9-(1-ethyl-1H-1,2,4-triazol-5-yl)-1-methyl-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
1-[(2-fluorophenyl)methyl]-4-(3-methoxypyrazin-2-yl)piperazin-2-one
(2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-{[(3-methylpyridin-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylic acid
3-(2-methanesulfonamidoethyl)-1-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-butyl-7-[(3-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(2R,3R)-3-amino-1'-[(3,5-dimethoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
3,5-dimethoxy-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}benzoic acid
3-(2,4-dimethoxybenzoyl)-1-(1-ethylpiperidin-4-yl)piperidine
6-(2,5-dimethylphenyl)-N-ethyl-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-4-azatricyclo[4.3.1.13,8]undecane
N-(2-aminoethyl)-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
1-[(3-fluorophenyl)methyl]-4-(1H-imidazol-2-ylmethyl)piperazine
2,5-dichloro-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzene-1-sulfonamide
2-cyclopropyl-9-(6-methoxypyrimidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecane
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}piperidine-1-carboxamide
2-{2-oxo-1'-[2-(pyridin-3-yl)acetyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-hydroxypyridine-3-carboxamide
2-methyl-4-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}phenyl)butan-2-ol
1-(4-chlorobenzoyl)-4-propyl-1,4-diazepan-5-one
8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-hydroxy-1-[3-(pyridin-2-yl)azetidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
2-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N,N-dimethylacetamide
2-{[methyl({[5-(oxan-2-yl)furan-2-yl]methyl})amino]methyl}-3,4-dihydroquinazolin-4-one
(1S,6R)-9-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
(2S,4R)-4-{4-[4-(2,3-dihydro-1H-isoindol-2-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
2-(3-fluoro-4-hydroxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
1-cyclohexanecarbonyl-4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-(3-ethoxybenzoyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine