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(3S,4R)-4-(3-methoxyphenyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine-3-carboxylic acid
2-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-6-(piperidin-3-yl)pyrimidin-4-amine
3-{[(4aS,8aR)-4a-(hydroxymethyl)-1-(pent-2-yn-1-yl)-decahydro-1,6-naphthyridin-6-yl]methyl}phenol
methyl 2-[4-({[(4-ethylphenyl)methyl](methyl)carbamoyl}amino)phenoxy]acetate
3-hydroxy-3-({[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
(4aS,8aR)-2-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-decahydroisoquinoline
7-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-(1H-indazol-6-yl)urea
5-(1-benzofuran-2-yl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1,2,4-triazin-3-amine
4-[6-(1-benzofuran-2-yl)pyrazine-2-carbonyl]morpholine
2-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-4-carbonitrile
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-methylpentane-1,2-dione
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
(1S,5R)-3-[(6-methoxy-2H-chromen-3-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(3-methylthiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}propanamide
2-chloro-4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
3-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1-(1-propyl-1H-1,2,3-triazol-4-yl)urea
3-hydroxy-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
2-chloro-N-methyl-5-[3-(1H-pyrazol-3-yl)phenyl]benzamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[(3-methyl-1-benzofuran-2-yl)methyl]cyclopentane-1,3-dicarboxamide
2-(3-hydroxypiperidin-1-yl)-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
9-(2-chloro-4-fluorobenzoyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl (2S,4R)-4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxylate
N-(furan-2-ylmethyl)-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
methyl[(1S)-1-phenylethyl]{[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}amine
2-ethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[2-(4-methoxyphenyl)ethyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
methyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
4-cyclobutanecarbonyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(pyrazin-2-yl)propan-2-yl]-1-(pyrimidin-2-yl)piperidin-4-amine
N-[4-(3-fluorophenyl)phenyl]-1-(oxane-4-carbonyl)piperidine-3-carboxamide
3-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(adamantan-1-yl)-5-(3-ethylmorpholine-4-carbonyl)pyrimidin-4-ol
2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-methoxy-6-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
N-({7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
5-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)methyl]-2-methoxyphenol
8-methyl-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]imidazo[1,2-a]pyridine-2-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
(3S,4S)-1-{[2-(2-hydroxyethoxy)phenyl]methyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[(3-methylphenyl)methyl]-1,4-diazepan-5-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,3,5-trimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(6-chloro-1,3-benzothiazol-2-yl)-N-(oxan-3-ylmethyl)piperidin-4-amine
3-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide