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N-({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
2-(2,3,6-trimethylquinoline-4-carbonyl)-1,2-oxazolidin-4-ol
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
6-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-[3-(2-fluorophenyl)benzoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-(dicyclopropylmethyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
1-{1-[1-(3,4-dimethoxyphenyl)propan-2-yl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
2-(3-{[4-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-indol-1-yl)acetamide
2-(pyridin-2-yl)-5-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}pyrimidin-4-ol
4-[(2-hydroxyethyl)sulfanyl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
2-benzyl-8-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
ethyl 3-[2-(4-butanamidophenyl)acetamido]butanoate
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(2-propoxyethyl)piperazine
methyl 2-chloro-4-{[(1-methyl-6-oxopiperidin-3-yl)carbamoyl]amino}benzoate
4-phenyl-1-{1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carbonyl}-1,2,3,6-tetrahydropyridine
4-methoxy-N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-N-(3-methylphenyl)benzamide
1-(1,2,3,4-tetrahydroquinolin-1-yl)-3-{[1-(thiophen-2-yl)propan-2-yl]amino}propan-1-one
N-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}thian-4-amine
3-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-6-methyl-3,4-dihydroquinazolin-4-one
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-3-methylfuran-2-carboxamide
3-[4-(3-cyanopyridin-2-yl)piperazin-1-yl]-N-[(4-methoxyphenyl)methyl]propanamide
4-(hydroxymethyl)-1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
benzyl(methyl)[(3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-oxazol-5-yl)methyl]amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
(1S,5R)-3-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(cyclopropylmethyl)-8-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}ethyl)-1H-indole
2-hydroxy-3-(2-methylphenoxy)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
5-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}-2-(3-methylphenyl)pyrimidine
3-(3-hydroxy-3-methylbutyl)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]benzamide
[1-ethyl-5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
(3S,4S)-4-(pyridin-2-yl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidine-3-carboxylic acid
1-benzyl-2-methyl-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
2-(3-methoxypropyl)-8-[3-(5-methylfuran-2-yl)butyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-{7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
[1-(1-cyclobutanecarbonylpiperidin-4-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
ethyl 4-[1-benzyl-3-(ethoxycarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine-1-carboxylate
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
2-amino-6-(2-amino-5-methyl-1,3-thiazol-4-yl)-4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]pyridine-3-carbonitrile
1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-3-[(dimethylamino)methyl]pyrrolidin-3-ol
4-({2-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2H-1,3-benzodioxol-5-yl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-[4-methyl-2-(pyrimidin-5-yl)phenyl]propanamide
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
(2S)-2-amino-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-phenylethan-1-one
3-butyl-1-methyl-4-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)piperazin-2-one