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2-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-methyl-1H-pyrazole
1-(1-cyclohexanecarbonylpiperidin-3-yl)-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-({2-[1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)-1H-pyrazole
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-methyl-4-(5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}furan-2-yl)but-3-yn-2-ol
N-{[4-(methylsulfanyl)phenyl]methyl}-N-propyl-3-(4H-1,2,4-triazol-4-yl)benzamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-methyl-1H-imidazol-1-yl)propanamide
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrrol-2-yl)propan-1-one
1-methyl-1'-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-(2-methoxyphenyl)-2-methyl-1-(1-propyl-1H-pyrazole-5-carbonyl)piperazine
1-(3-{4-[1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]pyridin-2-yl}phenyl)ethan-1-one
4-(2,2-dimethylcyclopropanecarbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(1H-pyrazol-1-yl)propyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
7-fluoro-3-({2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,2-dihydroquinolin-2-one
3-fluoro-5-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-[2-(dimethylamino)ethyl]-2,3-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-indole-7-carboxamide
2-fluoro-N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)benzamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}propan-1-one
3-({4-[1-(butane-1-sulfonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
2-[5-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
7-fluoro-2-methyl-4-[4-(oxolane-2-carbonyl)piperazine-1-carbonyl]quinoline
4-[5-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]benzamide
4-(hydroxymethyl)-1-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]piperidin-4-ol
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-1-phenylmethanesulfonamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
2-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyrazine
3-ethyl-1-[2-(ethylsulfanyl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]urea
(4aS,8aS)-2-(4,7,8-trimethylquinolin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
3-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1-propylurea
2-fluoro-N-{[3-(propan-2-yloxy)phenyl]methyl}-5-sulfamoylbenzamide
6-(hydroxymethyl)-N-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-1,4-oxazepane-4-carboxamide
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[2-(3-phenylpiperidin-1-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
4-methyl-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-imidazole-2-carboxamide
(2S,4R)-1-(3-methylbut-2-en-1-yl)-N-(propan-2-yl)-4-[3-(thiophen-2-yl)propanamido]pyrrolidine-2-carboxamide
5-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-ethylpyrimidin-2-amine
N-({4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
2-methyl-4-(4-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenyl)butan-2-ol
N-[(3-methyloxetan-3-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
1-(cyclopropylmethyl)-2-oxo-3-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
3-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenol
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
1-(cyclohexylmethyl)-N-[(3-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
8-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1-methyl-1H-imidazol-2-yl)({1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl})methanol
N-cyclopropyl-4-methoxy-2-{[1-(oxan-4-yl)piperidin-4-yl]oxy}benzamide
N-[3-(1H-imidazol-1-yl)propyl]-2-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)acetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,6-dimethylpyrimidine-4-carboxamide