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N-[3-(2-chlorophenoxy)propyl]-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-cyclohexyl-N3-methyl-N5-[(4-methylphenyl)(pyridin-4-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-(1H-imidazol-2-yl)-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidine
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-(3-methoxypropyl)piperidine
N-[(4-acetylmorpholin-2-yl)methyl]-2-(pyridin-3-yloxy)acetamide
methyl 3-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}benzoate
3-[3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
methyl 1-benzyl-5-{[1-(methylsulfanyl)propan-2-yl]amino}-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-{4-[(3-chloro-4-propoxyphenyl)methyl]piperazin-1-yl}-6-methylpyrimidin-2-amine
1-benzyl-8-[(4-fluorophenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-4-[2-(2-ethylphenoxy)ethyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
methyl 4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}benzoate
4-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(5-methylthiophen-2-yl)sulfonyl]-decahydro-1,6-naphthyridin-2-one
N-{3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-5-({[(3-phenoxyphenyl)methyl]amino}methyl)phenyl}acetamide
N-[3-(4-methylpiperazin-1-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
6-(3-ethoxyphenyl)-N4,N4-dimethylpyrimidine-2,4-diamine
3-(1-benzofuran-5-yl)-1-(3-methoxypropyl)-1-(1-methylpiperidin-4-yl)urea
N-[(3R,4R)-1-(2-chloro-4-fluorobenzoyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-(4-cyclopentylpiperazin-1-yl)-2-(3,4-dimethoxyphenyl)acetic acid
N-[(3R,4S)-4-cyclopropyl-1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]acetamide
4-{4-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2,6-dimethyl-4-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)phenyl acetate
1-[4-({[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
6-methyl-5-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(cyclobutylmethyl)-2-[(4-methylpiperazin-1-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
4-chloro-N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]pyrazine-2-carboxamide
3-chloro-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzene-1-sulfonamide
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-3-(N-methylmethanesulfonamido)propanamide
1-methyl-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]azepane-2-carboxamide
(2R)-2-amino-N-[1-(methoxymethyl)cyclopentyl]-2-phenylacetamide
N-cyclopropyl-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-({7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(dimethylamino)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}pyridine-3-carboxamide
1-ethyl-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
2-methyl-5-propyl-4-(4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazin-1-yl)pyrimidine
4-(6-ethylpyrimidin-4-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperazine-1-carboxamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
4-({ethyl[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]amino}methyl)-2,6-dimethylphenyl acetate
7-[(2,3-dimethoxyphenyl)methyl]-2-(2,2-dimethylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-methoxyethyl)-1-{1-[2-(trifluoromethyl)benzoyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide