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methyl (2S)-2-{[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-2-phenylacetate
3-cyclopropyl-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazole
7-(cyclopropylmethyl)-2-[2-(2-methylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-methyl-N-[4-({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}carbamoyl)phenyl]furan-3-carboxamide
N-(1-ethyl-1H-pyrazol-5-yl)-2-[4-(2-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)-1H-pyrazol-1-yl]acetamide
7-fluoro-3-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1-benzofuran-2-carboxamide
5-(1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
4-(1-ethylpyrrolidine-3-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(piperidin-1-ylmethyl)piperidine
N-benzyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
2-(2-chloro-4-fluorophenyl)-N-[(3-hydroxypyrrolidin-3-yl)methyl]acetamide
2-{1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-yl}benzoic acid
N,N-dimethyl-3-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]piperidine-1-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
7-(5-ethyl-1,2-oxazole-3-carbonyl)-N-(2-methoxyethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,4R)-1-(4-methoxy-2-methylbenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
1-(diphenylmethyl)-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-methoxy-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-2-phenylacetamide
4-[1-(2-carboxybenzenesulfonyl)piperidin-3-yl]benzoic acid
3-ethyl-5-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,2-oxazole
[(4-chloro-2-fluorophenyl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}propanamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-4-phenyl-1,2,3,6-tetrahydropyridine
2-(4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-1-yl)-1,3-benzothiazole
4-{5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-3-(4H-1,2,4-triazol-4-yl)propanamide
N-[2-(2,3-dichlorophenyl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
8-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
[(5-fluoro-2-methylphenyl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
3-({4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-(1-methyl-1H-pyrrol-2-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methanesulfonamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(pyridin-2-ylsulfanyl)propan-1-one
1-(4,5-dimethylthiophene-2-carbonyl)-N,N-dimethylazepan-4-amine
N-(6-hydroxy-6-methylheptan-2-yl)-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(1-{6-[butyl(methyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
2-amino-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-benzothiazole-5-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(1H-pyrazol-3-ylmethyl)benzamide
2-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}benzoic acid
3-(quinolin-8-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
2-benzyl-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(dimethyl-1,2-oxazol-4-yl)-N-(5-oxo-1-propylpyrrolidin-3-yl)acetamide
3-[2-oxo-2-(2-phenylmorpholin-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-(4-fluorophenyl)piperidin-3-amine