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N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-9H-purin-6-amine
N-(1H-indazol-7-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
3-({[2-(4-fluorobenzenesulfonyl)ethyl]amino}methyl)piperidin-3-ol
4-{[4-(4-butyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}-N,N-dimethylpiperazine-1-carboxamide
3-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
2-{2-[2-(dimethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}-N-(5-fluoro-2-methylphenyl)propanamide
3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-9H-purin-2-amine
(furan-2-ylmethyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(prop-2-yn-1-yl)amine
N-(2-chloro-5-methylphenyl)-3-oxa-9-azaspiro[5.5]undecane-9-carboxamide
{2-oxo-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}urea
N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-4-sulfamoylbenzamide
1-{2-[(4aR,8aR)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
2-(2-methoxyethyl)-9-[3-(4-methylphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-2-(pyridin-3-yloxy)acetamide
8-fluoro-3-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydroquinolin-4-one
N,N-dimethyl-3-[4-(piperidine-1-carbonyl)pyridin-2-yl]aniline
2-cycloheptyl-1-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
1-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-{1-methyl-1,4,9-triazaspiro[5.5]undecan-4-yl}ethan-1-one
5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N3-ethyl-N5-[(2-fluorophenyl)methyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(3R,5S)-5-(3-fluorophenoxymethyl)-N-(2-methylpropyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(5-oxopyrrolidin-2-yl)acetamide
5-{[(1S,5R)-3-[(dimethylcarbamoyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylfuran-2-carboxamide
N,N-dimethyl-5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-methyl-4-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-1,4-diazepane
4-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}azetidin-3-yl)pyridine
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(1,4-oxazepane-4-carbonyl)pyrrolidine-2-carboxylic acid
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]azepane
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dimethyl-1H-indol-5-ol
N-[(2-chlorophenyl)methyl]-2-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,3-oxazole-4-carboxamide
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[3-(pyridin-2-yl)propyl]benzamide
4-{5-methyl-2-oxo-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}benzonitrile
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]propanamide
ethyl({[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
1-{1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-2-yl}pyrrolidine
7-[(4-methoxy-2,5-dimethylphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(2R,3R,6R)-5-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-imidazol-1-yl)ethan-1-one
{4-[(2-chlorophenyl)methyl]-1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl}methanol
(2S,4S)-4-(4-chloro-2-methylbenzamido)-1-cyclopentyl-N-ethylpyrrolidine-2-carboxamide