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N,4-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
2-(dimethylamino)-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-4-(pyridin-3-yl)pyrimidin-2-amine
3-fluoro-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]oxane-4-carboxamide
5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-methoxy-1-{1'-[2-(methylamino)pyrimidine-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1'-[2-(1,2-benzoxazol-3-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-(1H-indole-3-carbonyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
3-amino-3-(3,4-dimethoxyphenyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
1-(1-cyclobutylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5-(2-fluorophenyl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
N'-{[2-(azepan-1-yl)-7-methoxyquinolin-3-yl]methyl}-N'-(furan-2-ylmethyl)-N,N-dimethylbutanediamide
3,6-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-{[2-(1-benzofuran-5-yl)-1H-imidazol-1-yl]methyl}-1-cyclopropanecarbonylpiperidine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-4-(1H-1,2,4-triazol-3-yl)benzamide
3-(1,3-benzothiazol-2-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
N-methyl-N-(pyrazin-2-ylmethyl)-3-(pyridin-3-yl)propanamide
N-[(1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperidin-4-yl)methyl]acetamide
N-[(4-fluorophenyl)methyl]-2-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)butanamide
2-[4-(2,1,3-benzothiadiazol-4-ylmethyl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
methyl 4-{[methyl({[1-(piperidin-1-yl)cyclohexyl]methyl})amino]methyl}-1H-pyrazole-3-carboxylate
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
(1S,4S)-5-(2,2-dimethylpropanoyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
5-(3-methylbut-2-en-1-yl)-1'-(oxolane-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-chloro-4-fluorophenoxy)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
4-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
3-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3,4-dihydropteridin-4-one
(2R,3R,6R)-5-(4-methyl-1,3-thiazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-methylpyridin-4-yl)-4-(2,4,5-trimethylbenzoyl)piperazine
1-[1-(propan-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-(5-methyl-2H-1,2,3-triazole-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(1-methyl-1H-pyrrole-2-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-1-methyl-N-(pyridin-4-ylmethyl)piperidine-2-carboxamide
[(3-chloro-4-methoxyphenyl)methyl](methyl)(pyrazin-2-ylmethyl)amine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
4-(3,5-dichloro-2-methoxybenzoyl)piperazine-2-carboxylic acid
N-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-N-methyloxolan-3-amine
N-[(3R,4S)-1-(4-methoxypyrimidin-2-yl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(6-methylpyridazin-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane