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4-[(1-acetylpiperidin-4-yl)oxy]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-methoxybenzamide
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,2,2-trimethylpiperazine
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-{[7-oxo-4-(2-oxo-2-phenylacetyl)-1,4-diazepan-1-yl]methyl}benzoate
5-{2-[4-(2-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
1-[(5-cyclopentylthiophen-2-yl)methyl]-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidin-2-one
[2-(diethylamino)-2-(furan-2-yl)ethyl][(5-methylfuran-2-yl)methyl]amine
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylacetamide
8-fluoro-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-2-carboxamide
ethyl 1-{3-[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]-6-(4-methylthiophen-2-yl)pyridin-2-yl}piperidine-4-carboxylate
1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-(morpholin-3-yl)ethan-1-one
(3R,4R)-3-cyclobutyl-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-methylpyrrolidin-3-ol
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
3-chloro-N-{[1-(cyclohex-2-en-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}benzamide
[(1-benzylpiperidin-4-yl)methyl](methyl){[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(1S,5R)-1,3,3-trimethyl-6-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-6-azabicyclo[3.2.1]octane
1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-(2-methylbutyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-(dimethylamino)-3-(4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperazin-1-yl)propan-2-ol
2-cyclopropyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(1R,2R,6S,7S)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
3-(2,6-dimethoxypyridin-3-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
5-(3,4,5-trimethoxyphenyl)-1H-indazole
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-N'-[2-(propan-2-yl)phenyl]butanediamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)azepan-2-one
3-[4-(6-methoxypyridin-3-yl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
1-ethyl-5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-1,2,4-triazole
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
2-(pyridin-2-yl)-5-{[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
2-methyl-N-[1-(thian-4-yl)piperidin-4-yl]-1-benzofuran-7-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(2-amino-1,3-thiazol-4-yl)propanamide
2-methyl-2-{4-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]phenyl}propanenitrile
N-[2-(2,4-dimethylphenoxy)ethyl]-2-(4-ethylpiperazin-1-yl)-N-methylacetamide
5-cyclobutanecarbonyl-1'-(4-methyl-1H-imidazole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cycloheptyl-3-methanesulfonamido-N-methylpropanamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(piperidin-3-yl)benzamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-chloro-N-cyclopentyl-4-{[1-(2-hydroxyethyl)piperidin-4-yl]oxy}benzamide
N-(3,4-dimethylphenyl)-3-(3-methylthiophene-2-carbonyl)piperidine-1-carboxamide
2-({4-[2-(propan-2-yl)-1H-imidazol-1-yl]phenyl}sulfanyl)acetamide
8-fluoro-2-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}quinoline
3-(4-methyl-1,3-thiazol-5-yl)-N-[(1R)-1-phenylethyl]propanamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-6-methylimidazo[1,2-a]pyridine-2-carboxamide
6-oxo-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
4-(5-ethylfuran-2-yl)-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one