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(1R,3S)-7-(3-chlorothiophene-2-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
(1S,2R)-2-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)amino}cyclohexan-1-ol
5-[3-(ethoxycarbonyl)pyridin-2-yl]thiophene-2-carboxylic acid
(isoquinolin-5-ylmethyl)(methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-[2-(2,6-dimethoxyphenoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
(3S,5R,9R)-5-hydroxy-11-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
(1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
9-(2-hydroxybenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]-N-(thiophen-2-ylmethyl)acetamide
(1S,2R)-2-{[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)amino}cyclohexan-1-ol
N-{2-[(2S)-2-acetamidopropanamido]-4-methylphenyl}benzamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)propanamide
3-(2-chloro-4-fluorophenyl)-5-(cyclopropylsulfamoyl)benzoic acid
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
4-[(4-fluorophenyl)methyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidine
N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(thian-4-yl)piperidine-4-carboxamide
4-(4-fluorophenyl)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-4-ol
1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-(5-methylfuran-2-yl)-1H-imidazole
(1S,3R)-3-amino-N-[2-(2-fluorophenoxy)pyridin-3-yl]cyclopentane-1-carboxamide
(4aS,8aR)-6-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-[4-(aminomethyl)benzoyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-6-ol
[(3R,5R)-5-[(dimethylamino)methyl]-1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]methanol
8-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}quinoline
1-[5-({[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
5-[3-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-5-propyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3,4-oxadiazole-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
8-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methylphenyl)ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(2-fluorobenzoyl)pyrrolidin-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
(3-{5-[2-(pyridin-3-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
1,4-dimethyl-9-{[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]azetidine-2-carboxylic acid
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(1S,9S)-11-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1-(morpholin-4-yl)cyclohexane-1-carboxamide
2-(dimethylamino)-N-[(4-hydroxyphenyl)methyl]-2-(4-methylphenyl)acetamide
3-methyl-7-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
5-chloro-N-(2-hydroxyethyl)-4,6-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(2,2-dimethyl-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}propyl)morpholine
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
ethyl (4aS,8aR)-6-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-decahydro-1,6-naphthyridine-4a-carboxylate
3-{2-[(2-hydroxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
6-[(diethylamino)methyl]-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-(hydroxymethyl)-1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidin-3-ol