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2-amino-4-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}quinazoline-6-carboxylic acid
1-(1-benzylpiperidin-4-yl)-N-[(3-methyloxetan-3-yl)methyl]piperidine-3-carboxamide
N5,N5-dimethyl-N6-[(4-phenyl-1,3-thiazol-5-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(3S,5R)-1-(3,5-dimethylbenzoyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
5-[(4-benzylpiperidin-1-yl)methyl]-N-(2-hydroxybutyl)-1,2-oxazole-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(1,2-thiazole-5-carbonyl)piperidine
3-methyl-5-[2-(4-methylphenoxymethyl)furan-3-yl]-1H-1,2,4-triazole
2-(3-{[2-(2-aminoethyl)quinazolin-4-yl]amino}propyl)phenol
1-(4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
(3aR,6aR)-2-[(3-chlorophenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1,3-oxazole-5-carboxamide
3-[(1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(3R,4S)-4-(3-methoxyphenyl)-1-(5-methyl-2-phenylfuran-3-carbonyl)pyrrolidin-3-amine
5-ethyl-N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}-1,2-oxazole-4-carboxamide
7-(3-chlorothiophene-2-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(2-methylphenyl)-3-(2-oxo-2-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethyl)-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
3-chloro-N-cyclopentyl-4-{[1-(pent-4-enoyl)piperidin-4-yl]oxy}benzamide
2-(3-methoxyphenyl)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidine
3-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-methyl-8-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-methyl-5-[4-(morpholin-4-yl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
[(1-cyclopentylpiperidin-4-yl)methyl]({[2-(prop-2-en-1-yloxy)phenyl]methyl})(pyridin-3-ylmethyl)amine
N3-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)piperidine-1,3-dicarboxamide
1-(2-{[(cyclopropylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
2-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]benzonitrile
2-(3-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}phenoxy)acetamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,6-difluorobenzamide
3-[1-(cyclohex-1-en-1-ylmethyl)-1H-imidazol-2-yl]phenol
4-{1-[1-(1H-imidazole-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-[(2R,3R)-2-methoxy-1'-(1,2,5-thiadiazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-4-(2-oxopyrrolidin-1-yl)butanamide
3-[3-(2-methoxyphenoxy)azetidin-1-yl]-6-methylpyridazine
N-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
(3S,4S)-1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-(piperidin-1-yl)pyrrolidin-3-ol
4-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperazine-2-carboxylic acid
N-[2-(3-methylpyridin-2-yl)ethyl]-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
N-[(2S)-2,3-dihydroxypropyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
2-methoxy-3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
3-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
3-benzyl-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-1,2-oxazole-5-carboxamide