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2,6-dimethyl-7-[4-phenyl-1-(1H-1,2,4-triazol-5-ylmethyl)-1H-imidazol-5-yl]heptan-2-ol
4-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-1-(4-methylphenyl)piperazin-2-one
2-hydroxy-N-[1-(pyrrolidine-1-carbonyl)azepan-3-yl]pyridine-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
7-(2-phenoxybenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-cyclobutyl-1-[6-hydroxy-4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-(ethylamino)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylpyrimidine-5-carboxamide
{5-[(1-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}piperidin-4-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
(2S,4S)-4-amino-1-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
8-[(2E)-2-methylbut-2-en-1-yl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 3-[(2-methylphenyl)methyl]-1-(oxan-4-yl)piperidine-3-carboxylate
2-cyclopentyl-N-[3-(4-{[3-(1H-imidazol-1-yl)-1-phenylpropyl]amino}piperidin-1-yl)phenyl]acetamide
4-(4-chlorophenyl)-N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)butanamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-4-(2-oxopyrrolidin-1-yl)benzamide
2-[({[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}amino)methyl]-5,8-dimethylquinolin-4-ol
3-(2-{2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-{[2-(3-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-2-methylpropanamide
(5-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}-2-(propan-2-yloxy)phenyl)methanol
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-1,3-thiazole-4-carboxamide
methyl 3-(1H-indol-3-ylmethyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-[(adamantan-2-yl)amino]-2-methylheptan-2-ol
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]propanamide
4-benzyl-3-[1-(oxane-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-{6-[(3-hydroxypropyl)(methyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
1-(2-acetamidoacetyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
2-benzyl-N-[2-(1H-indol-3-yl)ethyl]-1-methyl-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
(1S,5R)-3-(morpholine-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 2-[1-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
3,4,4-trimethyl-1-(5-methyl-4-phenylthiophene-3-carbonyl)pyrrolidin-3-ol
methyl 3-benzamido-5-({[5-(hydroxymethyl)furan-2-yl]methyl}amino)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl}-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
3-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
3-[({[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyrrolidin-3-ol
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(5-methanesulfonyl-2-methylphenyl)urea
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
(4aR,8aR)-2-[(2-chloro-5-fluorophenyl)methyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(2-methylpyrimidine-5-carbonyl)-decahydro-2,7-naphthyridine-2-carboxamide
[(6-methoxypyridin-3-yl)methyl](methyl)(1,3-thiazol-2-ylmethyl)amine
4-methyl-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,3-thiazole-5-carboxamide
(3S,4S)-4-cyclopropyl-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)pyrrolidine-3-carboxylic acid
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
2-(2-methoxyethyl)-9-[(4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
N-(4-methoxy-2-methylphenyl)-3-{1-[4-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide