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N'-(adamantan-1-yl)-N-methyl-N-(2-methylprop-2-en-1-yl)propanediamide
2-[1-(3-chloro-2-methylphenyl)-5-cyclobutyl-1H-1,2,4-triazol-3-yl]acetamide
N,N-diethyl-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxyethyl)-N-methylacetamide
5-({4-phenyl-5-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}methyl)-1H-1,2,4-triazole
2-[2-(5-acetylthiophen-3-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-({2-[(4-fluorophenyl)methyl]morpholin-4-yl}methyl)-2-methoxybenzoic acid
1-[1-(3-hydroxybutyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
3-(4,4-difluoropiperidine-1-carbonyl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
[1-(2-{[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]amino}ethyl)piperidin-2-yl]methanol
N-{2-[2-(furan-3-yl)-1H-imidazol-1-yl]ethyl}-4-methylpyridin-2-amine
N-[2-(4-fluorophenyl)-1-{1-[4-(1H-indol-3-yl)butan-2-yl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
(3S,4S)-1-(1-aminocyclobutanecarbonyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
N-(3-benzylphenyl)-2-(2-acetamidoethyl)piperidine-1-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
(3S,4S)-4-cyclopropyl-1-[4-(pyrrolidin-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
2-[4-(propan-2-yloxy)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
[(3R,4R)-1-(3-chloro-4-fluorobenzenesulfonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
3-(1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
6-{2-[2-(propan-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}-1H-indazole
5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(naphthalen-1-ylmethyl)amine
N-[(5-chlorothiophen-2-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-[(3S,4R)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(1S,6R)-9-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-[8-(2,2-dimethylpropyl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[(2R)-oxolan-2-ylmethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2-(2-methoxyethoxy)acetamide
{3-[(4-fluorophenyl)methyl]-1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-3-yl}methanol
N,2,6-trimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}quinoline-4-carboxamide
2-[(4-chlorophenyl)methyl]-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3aR,6aS)-5-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
(1S,4S)-2-(3,4-difluorophenyl)-5-[3-(3-methoxyphenyl)propanoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl 2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}piperidine-1-carboxylate
N-methyl-N-(1-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)thiophene-2-carboxamide
4,4,4-trifluoro-3-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)butanoic acid
({1-[1-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)dimethylamine
2-(1H-pyrazol-1-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}butanamide
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
methyl (2S)-2-[(2-cyclopropyl-1,3-benzoxazol-6-yl)formamido]-2-phenylacetate
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amine
4-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-1-(2-methoxyphenyl)piperazin-2-one
1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}urea
N-cyclopropyl-1-[(1s,4s)-4-[3-(4-methylphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-(4-fluorophenyl)-1H-pyrazole
6-(3-fluorophenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(2,3-dimethylphenoxy)acetamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
1-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione