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5-cyclobutanecarbonyl-1'-(2,3-dihydro-1H-inden-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[1-(pent-4-enoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
2-{[2-(1-cyclopentanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
4-{[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}-1-propylpyrrolidin-2-one
4-phenyl-1-(quinoxaline-5-carbonyl)piperidine-4-carbonitrile
methyl 2-(1-{2-[(2-fluorophenyl)methyl]-1,3-benzoxazol-6-yl}-N-methylformamido)acetate
2-[(3,4-difluorophenyl)methyl]-8-(3-fluoropyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine-3-carbonitrile
(3S)-1-{5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-methyl-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
N,N-dimethyl-2-{[3-(pyridin-3-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(2-methoxyphenyl)propanamide
methyl 3-{3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]propanamido}thiophene-2-carboxylate
2-(3-methoxypropyl)-9-(pyrimidin-5-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-(1-methanesulfonylpiperidin-4-yl)-1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
(3R,4R)-4-cyclopropyl-1-[(3,5-dichloropyridin-4-yl)methyl]-3-methylpiperidin-4-ol
4-ethyl-3-({1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-chlorophenyl)methyl]-3-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)propanamide
1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]cyclopropane-1-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(quinolin-6-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(3-cyclopentylpropanoyl)-4-ethyl-1,4-diazepan-5-one
3-(2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-[4-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
4-[(1-acetylpiperidin-4-yl)oxy]-N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-3-methoxybenzamide
[(1-cyclopentylpiperidin-4-yl)methyl][(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](pyridin-3-ylmethyl)amine
3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
3-(hydroxymethyl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-3-ol
1-[(2,4-dichlorophenyl)methyl]-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
(2R,3R)-1'-(3-fluoropyridin-2-yl)-3-(2-methyl-1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-methylpyridine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-methyl-1H-indole
4-[5-(1-benzofuran-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]-1-methylpiperidine
3-(4-acetyl-1,4-diazepane-1-carbonyl)-4-fluorobenzene-1-sulfonamide
6-{[(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)amino]methyl}-1,4-oxazepan-6-ol
(3aS,6aS)-2-cyclopentyl-5-(2,5-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-carbamoylcyclohexyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
1,2-dimethyl-4-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazine
1-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-2-(furan-2-yl)ethane-1,2-dione
1-[(4-chlorophenyl)methyl]-N-(1-propylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
1-(4-{methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}piperidin-1-yl)ethan-1-one
N-({1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methyl)-1-methylcyclopropane-1-carboxamide
4-[(dimethylamino)methyl]-1-{[4-(furan-2-yl)phenyl]methyl}azepan-4-ol
2-[(4-fluorophenyl)methyl]-4-(1-methylcyclopropanecarbonyl)morpholine
5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
4-[3-(2,2,2-trifluoroethoxy)benzoyl]piperazine-2-carboxylic acid
1-[1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)piperidin-3-yl]pyrrolidin-2-one
2-methyl-4-{4-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]phenyl}but-3-yn-2-ol