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3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]benzamide
(4aS,8aR)-6-(1-benzofuran-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(1R,5R)-6-(cyclopropylmethyl)-3-(3-fluoropyridin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-phenylethyl)-1-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)benzoic acid
N-[(2,4-difluorophenyl)methyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-(2-chlorophenyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidine
8-methoxy-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(4-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
4-[4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carbonyl]-1-phenylpiperazin-2-one
3,5-dimethyl-4-(3,4,5-trimethoxyphenyl)-1H-pyrazole
1-(2-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[(2E)-3-phenylprop-2-en-1-yl]cyclopropanamine
N-[2-(4-fluorophenyl)ethyl]-6-(methoxymethyl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[2-(propan-2-yloxy)propanoyl]piperazin-2-one
4-ethanesulfonamido-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
1-cyclohexyl-N-[(4-methoxyphenyl)methyl]-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
[1-(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
2-methyl-6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N4-[3-(3-fluorophenyl)phenyl]-N1,N1-dimethylpiperazine-1,4-dicarboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(2-chlorophenyl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(propan-2-yl)propanamide
4-(4-methoxyphenyl)-N-(oxan-2-ylmethyl)-4-oxobutanamide
3-methyl-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(oxolan-3-ylmethyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-6-(hydroxymethyl)pyridine-2-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-{1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
1-(2,4-dimethylphenoxy)-3-[(thian-4-yl)amino]propan-2-ol
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyridin-2-yl)propan-2-yl]amine
(1S,5R)-3-benzyl-6-(2-ethoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,4-diazepan-5-one
4-(3-methylpyridin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline
3-benzyl-4-(3,5-difluoro-4-methoxybenzoyl)piperazin-2-one
N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-(1-methyl-1H-indazol-3-yl)-2-{4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrrol-2-yl)pyridine
5-[1-(2-phenylacetyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2R,6R)-10-methoxy-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(pyridin-3-yl)acetamide
N-(oxolan-3-ylmethyl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
1-[(2-hydroxy-5-methoxyphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
dimethyl(2-{2-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-{[7-(cyclohex-3-en-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenoxyacetamide
2-[2-(3-chlorophenoxy)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-[3,5-bis(trifluoromethyl)phenyl]-N-(butan-2-yl)-4-hydroxy-N-methylpyrimidine-5-carboxamide
N-[1-(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide