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1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(3,4-dimethoxyphenyl)propan-1-one
1-cyclohexyl-N3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-methoxyethyl)-N-(propan-2-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}methanol
3-(5-{[(3-phenylprop-2-yn-1-yl)(propyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-(oxolane-2-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(4-ethoxyphenyl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
9-[(3-hydroxy-4-methoxyphenyl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]({[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})methylamine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-pyrazol-1-yl)propan-1-one
3-benzyl-7-{imidazo[1,2-a]pyrimidine-2-carbonyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
(1S,4S)-2-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}-2-azabicyclo[2.2.1]heptane
(4aS,8aR)-1-(2-aminoethyl)-6-(6-chloroquinolin-4-yl)-decahydro-1,6-naphthyridin-2-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]benzamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
2-methoxy-5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
3-({1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]azetidin-3-yl}oxy)pyridine
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(pyridin-3-ylmethyl)acetamide
[4-(2-phenoxyethyl)-1-(quinolin-2-ylmethyl)piperidin-4-yl]methanol
4-acetyl-N-(3-cyanophenyl)-4-phenylpiperidine-1-carboxamide
ethyl 2-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
9-(3-fluoropyridine-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
ethyl 4-(cyclopropylmethyl)-1-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]piperidine-4-carboxylate
3-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
2-(methylsulfanyl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
(1S,5R)-3-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
methyl 5-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(piperidin-3-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
6-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
N-[2-(4-fluorophenyl)-1-[1-(2-phenoxyacetyl)piperidin-4-yl]ethyl]-2-methoxy-N-methylacetamide
1-[1-(methoxymethyl)cyclobutanecarbonyl]-N-phenylpiperidin-3-amine
2,4-dimethyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[2-(pyrrolidin-3-yl)benzoyl]piperazine
1-(1,4-dioxan-2-ylmethyl)-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(3-acetylphenoxymethyl)-N-[(5-ethylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
5-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[1-(4-methyl-1,3-thiazol-2-yl)piperidin-4-yl]-2-phenylethan-1-ol
6-(pentafluoroethyl)-2-[2-(piperidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-(furan-3-ylmethyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-(3-phenylphenyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
4-methoxy-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
(1S,5R)-3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N-methylethane-1-sulfonamide