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1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
5-cyclopropyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2,2-dimethylpropan-1-one
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N4-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-({3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
methyl 5-(cyclohexylamino)-3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(2-amino-3-cyano-6-cyclopropylpyridin-4-yl)-N-methylbenzene-1-sulfonamide
4-[6-(propan-2-yl)pyridin-2-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[(dimethylamino)methyl]-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)pyrrolidin-3-ol
4-methyl-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-7-(methylsulfanyl)quinoline
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(3-methoxyphenyl)piperidine
5-[5-(2-propyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(1,3-thiazol-2-yl)piperazine
N-(butan-2-yl)-3-oxo-N-(thiophen-3-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
N-methyl-2-{1-[(2E)-2-methylpent-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
2-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxaspiro[4.4]nonan-2-one
4-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-ethylpiperazin-2-one
N-methyl-N-propyl-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-{2-[2-(1-benzothiophen-2-yl)-1H-imidazol-1-yl]ethyl}-6-methyl-3,4-dihydropyrimidin-4-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(3-ethoxy-2-hydroxypropyl)-5-methoxybenzamide
N-[(2R,3R)-2-ethoxy-1'-(2-oxo-2H-chromene-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-oxo-N-[2-(piperidin-1-yl)ethyl]propanamide
4-({[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
1-[(3S,4R)-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
4-{3-[3-cyclopentyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propyl}morpholine
3-(2-phenylethyl)-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
1-(2-chlorobenzoyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
1-[3-(2-methylpyrimidin-4-yl)phenyl]-N-(thiophen-3-ylmethyl)piperidin-4-amine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidine-3-carboxylate
4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-5-propylpyrimidine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
3-{[(2-hydroxy-3-methoxyphenyl)methyl](methyl)amino}-N-methylbutanamide
2-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(3-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-oxo-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[2-(1H-indazol-3-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(5-methylpyrazin-2-yl)methyl]benzamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]pyridine-3-carbonitrile
1-(1,3-benzoxazol-2-yl)-N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]piperidin-4-amine
N4-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-6-methylpyrimidine-2,4-diamine
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]urea