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N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-methyl-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N,N-dimethyl-3-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propanamide
(5-{[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}furan-2-yl)methanol
7-cyclopropanecarbonyl-N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(2-ethyl-1H-imidazol-1-yl)-N-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[6-(1-hydroxyethyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-N-phenylpropanamide
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrazine-2-carboxamide
1-(5-propyl-1,2-oxazole-3-carbonyl)-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}propan-1-one
2-({2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)acetamide
4-(piperidin-3-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}benzamide
1-{[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
[(2-chloro-4,5-diethoxyphenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-(3-propoxypiperidin-1-yl)-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
N-{2-[(3-ethyl-5-hydroxyadamantan-1-yl)formamido]ethyl}pyridine-3-carboxamide
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(pyrimidin-4-ylmethyl)-1H-pyrazole-3-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-butyl-4-phenyl-1H-imidazol-1-yl)propan-1-ol
N-[(2-fluorophenyl)methyl]-2-[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
[(5-{1-[(4-tert-butylphenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
3-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-ethyl-1H-pyrazole
N-methyl-N-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]cyclohexanamine
1-[2-methoxy-4-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
5-[4-(1-ethoxyethyl)phenyl]pyrimidine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
(3S)-1-[3-(1H-imidazol-2-yl)benzoyl]pyrrolidin-3-amine
1-(3-methoxybenzenesulfonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
(1R,5R)-6-benzyl-3-(3-fluoropyridin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-(4-methylphenyl)-5-(pyrimidin-5-yl)-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)azepane-1-sulfonamide
N-(4-fluoro-3-methylphenyl)-3-[2-(4-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propanamide
1-[(3-chloro-5-fluorophenyl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-5-methyl-1,3,4-oxadiazol-2-amine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
N-cyclopropyl-1-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]piperidine-3-carboxamide
3-(2-fluorophenyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylpropanamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
[3-(cyclopropylmethyl)-1-(2-methylfuran-3-carbonyl)piperidin-3-yl]methanol
methyl 4-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-4-oxobutanoate
2-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)methyl]-5,8-dimethylquinolin-4-ol
3,5,7-trimethyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-indole-2-carboxamide
2-[3-methyl-5-(3-phenoxypropyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)oxane-4-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2H-1,3-benzodioxole-5-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-cyclobutylpiperidine-4-carboxamide
(1R,5R)-6-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide