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4-(4-methoxy-3-methylphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(2-fluorophenyl)methyl]-2-{[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]amino}acetamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
5,6-dimethyl-3-(pyridin-3-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(4-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}acetamide
(3aR,7aS)-N-(3-fluoro-4-methylphenyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
(2S,4S,5R)-4-[(2-carboxyethyl)carbamoyl]-2-ethyl-5-(4-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-[2-(methylsulfanyl)benzoyl]piperidine
ethyl 2-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]acetate
1-amino-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}cyclopentane-1-carboxamide
2-(1-propylpiperidin-4-yl)-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
(3S,4R)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
(3S,4R)-4-(3-methoxyphenyl)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-(2-{4-[(1-phenyl-1H-pyrazol-5-yl)methyl]morpholin-2-yl}ethyl)acetamide
N-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
1-{4-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-(adamantan-2-yl)-4-[(2S,4S)-1-benzyl-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]piperazine
1-{3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}ethan-1-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-(3-methoxypropyl)-8-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-(cyclohex-3-ene-1-carbonyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)(1,3-thiazol-4-ylmethyl)amine
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
3-({7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenol
1-methyl-4-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)piperazine-2-carboxylic acid
1-[3-(methoxymethyl)piperidin-1-yl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
(3S,4S)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(3S,4S)-4-cyclopropyl-1-[2-(methylamino)pyridine-3-carbonyl]pyrrolidine-3-carboxylic acid
1-methyl-6-oxo-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,6-dihydropyridazine-3-carboxamide
methyl 5-oxo-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]pentanoate
1-ethyl-N-[(2-fluorophenyl)methyl]-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(4aR,7aS)-4-(2-ethoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-one
(1R,3S)-N-[(4-fluorophenyl)methyl]-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}pyridine-4-carboxamide
(2R)-2-hydroxy-1-[4-(2-methylphenoxy)piperidin-1-yl]-2-phenylethan-1-one
4-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-imidazol-2-yl}-2-methyl-1,3-oxazole
3-[4-(2-methoxyphenoxy)piperidin-1-yl]-N-(pyridin-3-yl)propanamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[4-(methylsulfanyl)benzoyl]piperidine
N-[(3S,4R)-1-(2-hydroxypyridine-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-[(3-methoxyphenyl)methyl]-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-({1-[(3-cyanophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)thiophene-2-carboxamide
2-[2-oxo-1'-(thiophene-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
4-(1H-imidazol-2-yl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
1-benzyl-8-{[5-(hydroxymethyl)furan-2-yl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)thiophene-2-carboxamide
N,N-dimethyl-1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidin-3-amine