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(2S,4S,5R)-4-[(carboxymethyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[(3-{[(1S)-1-phenylpropyl]carbamoyl}phenyl)amino]acetic acid
1-(2-oxo-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
1-(3-methoxyphenyl)-3-methyl-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
4-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
2-[6-(pyrrolidin-1-yl)pyridazin-3-yl]benzoic acid
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[2-(4-methylpiperidin-1-yl)ethyl]amino}methyl)piperidin-2-one
N-(cyclohex-3-en-1-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(3-methylbutanoyl)piperidine-2-carboxamide
N-methyl-4-[5-(piperidin-1-ylmethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
9-[(3-chloro-4-methoxyphenyl)methyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]methylamine
1-(2-methylbenzoyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-cyclooctyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methyl-1,3-benzothiazole-5-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3-methoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-methylpyrimidin-4-amine
3-(1,3-benzothiazol-2-yl)-1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}propan-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,N-diethyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(quinolin-8-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(dimethylamino)-N-(3-ethoxypropyl)-2-(3-methylphenyl)acetamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]acetamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3,4,5-trimethoxyphenyl)methyl]amine
4-[(3R)-3-hydroxypyrrolidin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
1-phenyl-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2,6-dimethoxybenzamide
6-[3-(oxan-4-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
4-[(4-{3-[4-(propan-2-yl)piperidine-1-carbonyl]piperidin-1-yl}piperidin-1-yl)methyl]pyridine
1'-[(3-fluorophenyl)methyl]-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{5-[2-(dimethylamino)phenyl]-1H-indazol-1-yl}acetamide
1-tert-butyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrrolidin-2-one
N-(5-oxo-1-phenylpyrrolidin-3-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
(4aS,8aR)-1-(3-methoxypropyl)-6-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
(3R,4R)-4-{[4-(3-chlorophenyl)pyrimidin-2-yl]amino}piperidin-3-ol
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]amine
7-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[5-(2,4-difluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2-(methoxymethyl)piperidine
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-(4-methoxyphenyl)butan-1-one
N-(3-methoxyphenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methylpyrazolo[1,5-a]pyridine-7-carboxamide
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(pyridazine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 2-(2-{2-[4-(4-oxo-4-phenylbutanamido)-1H-pyrazol-1-yl]acetamido}ethyl)-1,3-thiazole-4-carboxylate
N-methyl-N-[2-(methylsulfanyl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-(pyridin-4-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propane-1,3-diol
5-{[benzyl(methyl)amino]methyl}-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide