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1-cyclopropyl-5-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]piperidin-2-one
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(2,1,3-benzoxadiazol-5-ylmethyl)methylamine
1-(3,5-dimethylphenyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperazin-2-one
methyl 6-(2-benzyl-3-oxopiperazine-1-carbonyl)pyridine-3-carboxylate
4-[(3-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)methyl]morpholine
5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1-[2-(thiophen-2-yl)ethyl]-1H-imidazole
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-methyl-6-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
(2R)-N-[3-(1H-imidazol-1-yl)propyl]-2-phenyl-N-(pyridin-4-ylmethyl)butanamide
1-[4-(4-{[(1R,2S)-2-(methoxymethyl)cyclopentyl]amino}piperidin-1-yl)phenyl]-3-methylimidazolidin-2-one
1-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(3-fluoro-4-methoxyphenyl)benzamide
1-[2-(1-benzothiophen-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(6-hydroxy-6-methylheptan-2-yl)piperidine-3-carboxamide
N-(2-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
6-(methoxymethyl)-N,1-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclopropyl-2,7-dioxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3-diazepane-4-carboxamide
1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
benzyl(oxolan-3-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
4-chloro-N,N-dimethyl-5-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}-1,3-thiazol-2-amine
1-(carbamoylmethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
1-[(1-ethylpiperidin-3-yl)methyl]-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
1-cyclopropanecarbonyl-4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}piperidine
(3R,4S)-4-cyclopropyl-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}pyrrolidin-3-amine
N-ethyl-3-(4-fluorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenylpropanamide
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-3-propyl-1H-pyrazole-5-carboxamide
methyl (2S,4R)-4-(dimethylamino)-1-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]pyrrolidine-2-carboxylate
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}pyrimidine-5-carboxylic acid
1-{3-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}imidazolidin-2-one
4-[(cyclopropylmethyl)amino]-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
N3-[2-(3-fluorophenyl)ethyl]-N5-[3-(methylsulfanyl)propyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
6-ethyl-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-methylquinoline-4-carboxamide
2-methoxy-1-{1'-[(2S)-pyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-(methoxymethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]cyclobutane-1-carboxamide
3,4-difluoro-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzene-1-sulfonamide
2-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
2-{2-[(1,4-dithiepan-6-yl)amino]ethyl}-3,4-dihydroquinazolin-4-one
N'-(2,4-dimethylphenyl)-N-(1H-imidazol-2-ylmethyl)propanediamide
(3aS,6aS)-2-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]propane-1,2-diol
1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(morpholin-2-yl)ethan-1-one
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-({[4-(propan-2-yl)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-(prop-2-en-1-yl)-9-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-fluorophenoxy)piperidine
1-cyclohexyl-4-[3-(3-methoxyphenyl)propanoyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-(2-fluoro-4-methylbenzoyl)-3-(2-methylphenoxymethyl)piperidine
1,4-dimethyl-9-(3-propyl-1H-pyrazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecane
6-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]pyridine-2-carbonitrile
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one