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({4-ethyl-5-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N-(3-hydroxypropyl)piperidine-3-carboxamide
9-(2,3-dihydro-1H-indene-1-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-methoxy-5-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
2-(dimethylamino)-2-(2-fluorophenyl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
4-[1-benzyl-5-(2-methyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-[2-(3-hydroxy-3-methylpiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-phenylpyrrolidin-3-ol
(1R,2R)-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-2-phenylcyclopropane-1-carboxamide
1-(2-ethoxyacetyl)-4-(pyrazin-2-yl)-1,4-diazepane-6-carboxylic acid
(1S,4S)-5-[(4-chlorophenyl)methyl]-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-4-[(2-hydroxyethyl)(propan-2-yl)carbamoyl]-1-methylpyrrolidine-2-carboxylate
5-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]pentan-2-one
3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]benzonitrile
1-(2-methoxyethyl)-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-1-(thiophen-3-ylmethyl)urea
3-ethyl-8-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-ethyl-1-[2-(4-phenylpiperazin-1-yl)ethyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(5R)-5-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
N-benzyl-N-methyl-3-(1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}piperidin-4-yl)propanamide
4-[4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperazin-1-yl]quinazoline
3-{[4-(methylamino)piperidin-1-yl]sulfonyl}-N-(oxolan-3-ylmethyl)benzamide
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridin-2-amine
1-(4-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)ethan-1-one
N-(3-methoxypropyl)-6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[5-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-2-methoxyphenyl]acetamide
8-methoxy-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)quinoline
5-ethyl-2-[3-methyl-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyridine
2-cyclopentyl-2-phenyl-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
3-{[(4-fluorophenyl)methyl]amino}-N-[(4-methoxyphenyl)methyl]-5-(pyrrolidine-1-sulfonyl)benzamide
N-[4-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)phenyl]acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-oxo-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-3-phenylpyrrolidine-2,5-dione
N-{2-[(3,4-dimethyl-5-sulfamoylphenyl)formamido]ethyl}pyridine-3-carboxamide
N-(2-hydroxyethyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N,N-dimethyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
2-(1-tert-butyl-1H-pyrrole-3-carbonyl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
3-{2-[({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
2-methoxy-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}acetamide
3-{1-[(1,2-dimethyl-1H-indol-3-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
methyl 4-{4-[3-(1H-imidazol-1-yl)butanoyl]piperazin-1-yl}benzoate
2-(2-aminoethyl)-N-[furan-2-yl(phenyl)methyl]quinazolin-4-amine
methyl (2S,4S)-1-[(2-methoxyphenyl)methyl]-4-(2-phenylquinoline-4-amido)pyrrolidine-2-carboxylate
6-(1H-pyrazol-3-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-(2-phenoxyphenyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}urea
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-ol
N,N-dimethyl-2-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]acetamide
N-{[1-(dimethylamino)cycloheptyl]methyl}pyrimidin-4-amine