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N-[(trimethyl-1H-imidazol-2-yl)methyl]quinoxaline-5-carboxamide
1-(4-{[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
2-{3-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]phenoxy}acetamide
1-propyl-4-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}pyrrolidin-2-one
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(2,2-dimethyloxan-4-yl)formamido]methyl}benzoate
3-[5-(ethanesulfonyl)thiophen-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
8-(2,6-dimethoxypyrimidin-4-yl)quinoline
1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-4-[2-(1,3-thiazol-4-yl)acetyl]-1,4-diazepan-2-one
2,6-di-tert-butyl-4-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]phenol
1-cyclobutanecarbonyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
8-(6-methylpyridazin-3-yl)-1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-1,8-diazaspiro[4.5]decane
1-[(4-ethylphenyl)methyl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-oxopyrrolidine-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
5-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1-(3-phenylpropyl)piperidin-2-one
1-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(4-methylphenyl)methyl]amine
(3S,4S)-1-[(2-ethylpyrimidin-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
1-ethyl-5-[ethyl(2-methylprop-2-en-1-yl)amino]-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-methoxypropan-1-one
3-({2-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-(propan-2-yl)-4H-1,2,4-triazole
N-propyl-6-(1H-pyrazol-4-yl)pyridine-3-carboxamide
(4aS,8aR)-6-(1H-indole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[benzyl(methyl)amino]-3-(4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)propanamide
1-{1-[3-(azepane-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperidin-4-yl}piperidin-4-ol
7-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidine
N-[(2R,3R)-2-methoxy-1'-[(2E)-4-methylpent-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-[4-(1,3-benzothiazol-2-yl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-hydroxybenzamide
2-[1-(2-methylpropyl)-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
6-[4-(1-methoxyethyl)phenyl]-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
(1R,3S)-3-ethoxy-7-(2-phenoxybenzoyl)-7-azaspiro[3.5]nonan-1-ol
1-phenyl-4-({2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)-1H-1,2,3-triazole
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4-methylpiperazine
N-cyclopropyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
N-cyclopropyl-5-(1H-imidazol-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
1-(2-amino-6-methylpyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(2-methoxyphenyl)-3-{1-[1-(3-phenylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[4-(butan-2-yl)phenyl]-4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carboxamide
2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]acetamide
3-{[(5-chloro-2-hydroxyphenyl)methyl]amino}-5-(dimethylsulfamoyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
2-(dimethyl-1,2-oxazol-4-yl)-2-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
5-(1,4-dioxane-2-carbonyl)-3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-cyclobutyl-3-{[(1-propyl-1H-imidazol-2-yl)methyl]sulfamoyl}benzamide
(4aR,8aS)-1-[3-(dimethylamino)propyl]-6-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1,2-dimethyl-5-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-imidazole
4-{methyl[(1-methylpyrrolidin-2-yl)methyl]amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
3-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-N-[(2-chlorophenyl)methyl]propanamide