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4-(hydroxymethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
4-(7-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)morpholine
4-[(2,6-difluoro-4-methoxyphenyl)methyl]-1-phenylpiperazin-2-one
4-benzyl-1-(4-methoxy-3-methylbenzoyl)piperidine-4-carboxylic acid
5-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-methyl-2-(methylamino)-N-{[1-(oxan-4-yl)piperidin-4-yl]methyl}benzamide
N-(2-methylpropyl)-2-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3,3-diphenylpiperidine
(1S,5R)-3-{[4-(difluoromethoxy)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
7-methyl-3-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
1-benzyl-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
{1-[2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]piperidin-2-yl}methanol
2-[(1S,5R)-3-(6-cyanopyridin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
5-chloro-N-(1,4-dioxan-2-ylmethyl)thiophene-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(2-oxopyrrolidin-1-yl)propanamide
(5S,9aS,9bS)-5-[5-(methoxymethyl)furan-2-yl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-(benzyloxy)-1-cyclohexyl-4-(pyridine-4-carbonyl)-1,4-diazepan-2-one
(3aS,6aS)-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{5-methyl-2-[2-(methylamino)ethoxy]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(3-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
N-(3,4-dimethoxyphenyl)-1-(4-methoxypyrimidin-2-yl)piperidin-3-amine
3-{5-[3-(hydroxymethyl)quinolin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-(4-{[3-(2-methylpropyl)pyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)-1-(oxan-4-yl)piperidine
N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
2-{3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-(furan-3-ylmethyl)-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-methyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-methoxyethyl)-1,2-oxazole-3-carboxamide
2-({[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}methyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-6-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-[(3S,4R)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[3-(4-methoxyphenyl)propyl]propanamide
(1-{[1-(3-methylbenzenesulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-(naphthalen-2-ylmethyl)-N-(2-phenylethyl)piperidine-3-carboxamide
N'-(5-chloro-2-methylphenyl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]propanediamide
2-cyclopropyl-N-(pyridin-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one
1-(1H-indol-2-ylmethyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
1-ethyl-4-(2-oxo-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)piperazine-2,3-dione
1-[2-(1-hydroxycyclopentyl)ethyl]-5-methyl-5-phenylpiperidin-2-one
6-(morpholin-4-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
(2R,3S,6R)-3-phenyl-5-[3-(1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}-3-(3-methyl-1H-1,2,4-triazol-5-yl)propanamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylpiperidin-4-yl)piperidine
2-ethoxy-5-{2-[(2-hydroxyethyl)(methyl)amino]pyrimidin-4-yl}benzoic acid