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[3-(6-chloro-1H-1,3-benzodiazol-2-yl)-2,4,6-trimethylphenyl]methanol
N-[4-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
ethyl 3,5-dimethyl-4-[methyl(quinolin-5-ylmethyl)carbamoyl]-1H-pyrrole-2-carboxylate
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-4-(4,4,4-trifluorobutanoyl)-1,4-diazepan-2-one
5-ethyl-2-methyl-N-[2-(morpholin-4-yl)ethyl]pyrimidin-4-amine
N-tert-butyl-3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(2-methoxyethyl)-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
N-(3-fluorophenyl)-N-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]methanesulfonamide
2-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-8-methoxyquinoline
N-{[3-(trifluoromethoxy)phenyl]methyl}oxolane-3-carboxamide
6-({[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}methyl)-N-[1-(naphthalen-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-(5-methyl-4-{[2-(thiophen-3-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]benzamide
2-cyclobutyl-1-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]ethan-1-one
(1S,5R)-6-methyl-3-[1-(4-methylphenyl)cyclopropanecarbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(pyridin-3-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidine-5-carboxamide
N-ethyl-5-{1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidin-2-amine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N'-(adamantan-1-yl)-N-[(2-methoxyphenyl)methyl]propanediamide
1-methyl-2-oxo-N-[1-(thiophen-3-yl)propan-2-yl]-1,2-dihydroquinoline-3-carboxamide
N-{2-[ethyl(methyl)amino]butyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-indol-1-yl)propyl]acetamide
7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-methyl-4-(5-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
3-[(3R,4S)-1-(furan-3-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-fluoro-N,6-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-N-(1-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propan-2-yl)aniline
4-methyl-2-oxo-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pentanamide
N-(3-fluoro-2-methylphenyl)-2-[(prop-2-en-1-yl)(prop-2-yn-1-yl)amino]acetamide
2-(2-hydroxyethyl)-9-(3-propyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-3-yl)methanol
methyl 5-[3-(3-methoxyphenyl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methyl-1H-pyrazole-4-carboxamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethyl-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N,N-dimethyl-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-sulfonamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]piperazine
3-[(dimethylamino)methyl]-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-3-ol
2-[4-(3-chloro-4-methoxyphenyl)-1H-pyrazol-1-yl]propanamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(2-hydroxyethyl)-3-(1-methylpiperidin-3-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
3-methyl-4-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}-1,2,5-oxadiazole
2-(isoquinoline-1-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
3-hydroxy-N-[4-(2-methoxyphenyl)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1-propyl-1H-pyrazole-5-carboxamide
N3-[3-(2,4-dimethylphenoxy)propyl]-N1,N1,N3-trimethylpiperidine-1,3-dicarboxamide
1-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methyl}-3-(propan-2-yl)urea