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2-methyl-4-{4-[(4-methyl-3-phenylpiperazin-1-yl)methyl]phenyl}butan-2-ol
2-[(adamantan-1-ylmethyl)[(2-methyl-1,3-oxazol-4-yl)methyl]amino]ethan-1-ol
N-cyclopropyl-3-{[2-(3-fluorophenyl)-2-hydroxyethyl]sulfamoyl}benzamide
N-[1-ethyl-2-(2-fluorophenyl)-7-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-5-yl]acetamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-ethyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-2-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-(oxolan-3-yl)benzamide
2-cyclopropyl-9-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-3-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}quinolin-4-amine
4-(1H-pyrazol-1-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine-4-carboxylic acid
1-{2-oxo-2-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethyl}-1,2-dihydroquinolin-2-one
5-methyl-N-[2-(piperidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopropyl-5-(3-hydroxybenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N,2-dibenzyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine-4-carboxylate
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-4-phenylbutane-1,2-dione
N-[3-(2-methoxyacetamido)-2-methylphenyl]azepane-1-carboxamide
{1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-3-[(3-chlorophenyl)methyl]piperidin-3-yl}methanol
(2S,4R)-4-amino-1-(2-methoxyquinoline-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(5-{[3-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-{2-[methyl({[2-(propan-2-yl)pyrimidin-5-yl]methyl})amino]ethyl}piperidin-2-one
5-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
N-(1H-1,2,4-triazol-3-ylmethyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(methoxymethyl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
(1S,5R)-3-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
4-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N-[3-(furan-2-yl)phenyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[(1-acetylpiperidin-4-yl)oxy]-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3-methoxybenzamide
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(5-ethylfuran-2-yl)pyridine-3-carbonitrile
2-(4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
N-methyl-3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperazine
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
1-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
3-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
(1R,4S)-1,7,7-trimethyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-2-methoxy-N-methyl-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(4-methoxyphenyl)propan-1-one
(2R,3R)-3-(2-methyl-1H-imidazol-1-yl)-1'-(pyridin-4-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(5-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]propan-1-one