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(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
5-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]-2-methoxyphenol
2-[benzyl({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
1-(2-phenylethyl)-8-(1-propylpiperidin-4-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-({[4-(3-fluorophenyl)oxan-4-yl]methyl}amino)-N-(pyridin-3-yl)propanamide
1-cyclopropanecarbonyl-4-[4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenoxy]piperidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-3-methylpiperidine
1'-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3-chlorophenyl)methyl]({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)acetamide
1-[1-(3-chlorobenzoyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-ol
4-fluoro-N-({1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}methyl)benzamide
2-(4-chlorophenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
4-(6-methyl-2-phenylpyrimidin-4-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
7-(cyclopropylmethyl)-2-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decane
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[(5-methylfuran-2-yl)methyl]pyrimidin-2-amine
3-methyl-N-{1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
4-{[(3R,4S)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]methyl}benzoic acid
(1S,5R)-6-(2-methoxyethyl)-3-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,3,4-trimethoxybenzamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[3-(3-carbamoylpiperidin-1-yl)propyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[(diethylamino)methyl]-5-ethyl-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]furan-2-carboxamide
N-[(2S)-1-[2-(azocan-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-1-oxopropan-2-yl]acetamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
5-(3-chlorophenyl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1,2,4-triazin-3-amine
6-methyl-4-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
(2S,4R)-4-{4-[4-(azepan-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
4-(1,4-oxazepane-4-carbonyl)-1,2-dihydrophthalazin-1-one
N-(2-methoxyethyl)-3-{[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]oxy}benzamide
4-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-1-cyclohexylpiperazin-2-one
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(2-methoxyethyl)-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]piperidine-3-carboxamide
9-(cyclopropylmethyl)-4-(4-fluorobutyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
1-[9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
benzyl (4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-(2-methoxy-4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-3-(pyrazin-2-yl)propan-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(2,4-dimethoxybenzoyl)piperidine
(3S,7S,8aS)-3-(2-methylpropyl)-7-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-(pyrrolidin-1-yl)-3-{1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-3-yl}propan-1-one
1,3-dimethyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-1H-pyrazole-5-carboxamide
4-[(2-ethoxyphenyl)methyl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one