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(2R,3R,6R)-5-(2-fluorobenzoyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
({5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-(3-fluoropyridin-4-yl)-4-(hydroxymethyl)piperidin-4-ol
2-(2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
(1S,5R)-6-(cyclobutylmethyl)-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-2-methoxyphenol
1-[2-(pyridin-2-yl)pyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
5,5-dimethyl-3-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,3-oxazolidine-2,4-dione
1-(furan-2-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S,5R)-4-(4-ethylpiperazine-1-carbonyl)-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-{3-[methyl(phenyl)amino]propyl}-3-propanamidobenzamide
ethyl 4-[4-hydroxy-2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperazine-1-carboxylate
3-(3-methyl-1H-pyrazol-1-yl)-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}propanamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-3-(3,4,5-trimethoxyphenyl)-1H-pyrazole
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(2-methylprop-2-en-1-yl)benzamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
N-ethyl-4-{[(oxan-3-ylmethyl)carbamoyl]amino}-N-phenylbenzamide
2-[2-(2,3-dimethylphenoxy)ethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-(1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
8-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
ethyl 4-({1-[4-(3-phenylpropanamido)phenyl]piperidin-4-yl}amino)piperidine-1-carboxylate
2-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]-1,2-oxazinane
3-[2-(methylsulfanyl)benzoyl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
4-({4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(3-methoxyphenyl)methyl](oxolan-2-ylmethyl)amine
4-(4-ethyl-1H-pyrazol-5-yl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidine
(1R,7S)-3-cycloheptyl-N-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1,3-dimethyl-6-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,5S)-1-benzyl-N-[(3,4-dimethoxyphenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
3-cyclopropyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-(2-methylpropyl)-6-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(1-hydroxy-2-methylpropan-2-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-chloro-4-fluoro-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
(3R,4S)-1-(7-chloroquinolin-4-yl)-4-cyclopropylpyrrolidin-3-amine
9-(2-hydroxyethyl)-1-methyl-4-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N-(1,3-thiazol-2-yl)propanamide
1-methyl-3-(2-methylpropyl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-fluoro-2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3,8-dimethylquinoline
(2S,4S)-4-amino-1-[(2-butyl-1H-imidazol-4-yl)methyl]pyrrolidine-2-carboxylic acid
N-{[1-(2-phenoxyacetyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
2-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
2-(cyclopropylmethyl)-9-({3-[(dimethylamino)methyl]phenyl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-N-ethyl-1-[(4-methoxy-2-methylphenyl)methyl]-4-(3-methoxypropanamido)pyrrolidine-2-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
7-(2-cyclohexylethyl)-2-(2-hydroxy-2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one