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N-[2-(furan-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
N-(1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
7-(4-chlorophenyl)-2-(5-methylpyrazin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(1R,3S)-7-(2H-1,3-benzodioxole-5-carbonyl)-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
1-(2-fluorophenyl)-4-[(4-{[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
(1S,3R)-N1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
8-(4-fluorobenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
(3R,5S)-5-(morpholine-4-carbonyl)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]piperidine-3-carboxamide
5-[1-(2-methylpropyl)pyrrolidin-2-yl]-N-(pyridin-3-yl)thiophene-2-carboxamide
N-[(4-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1-[6-(3-fluorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
2-{1-benzyl-4-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
[1-(cyclohexylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[4-(trifluoromethyl)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
N,N-dimethyl-2-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}benzamide
2-amino-4-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-methyl-4-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-3-(1-methyl-1H-pyrazol-5-yl)propanamide
4-(2-ethylpyrimidine-5-carbonyl)thiomorpholine
2-(3-fluorophenyl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
methyl 4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazine-1-carboxylate
N-cyclopropyl-5-(phenoxymethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
(2R,3R)-3-(dimethylamino)-1'-(3,5-dimethylfuran-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(6-hydroxypyrimidin-4-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(2-hydroxyphenoxy)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
3-(1-{1-[(3E)-pent-3-enoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)benzoic acid
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]propan-1-one
(2R)-2-{[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
6-methyl-N4-[1-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine
3-{4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N-{3-[2-(morpholin-4-ylmethyl)phenoxy]phenyl}acetamide
4-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
4-[(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)methyl]morpholine
4-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-1,2-dihydroquinolin-2-one
3-[(2R,3R,6R)-5-(furan-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-(methylamino)pyridine-3-carboxamide
N4-methyl-N4-(oxolan-2-ylmethyl)-6-(propan-2-yloxy)pyrimidine-2,4-diamine
2-methoxy-4-{[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N,N-dimethyl-2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}pyridine-3-carboxamide
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N'-(3,5-dimethylphenyl)-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]propanediamide
5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-{3-oxo-3-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propyl}imidazolidine-2,4-dione
5-{4-[1-hydroxy-2-(morpholin-4-yl)ethyl]phenyl}thiophene-2-carboxylic acid
N-[2-(1H-indol-1-yl)ethyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide