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3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-[(3-methoxyphenyl)methyl]piperidine
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-2-(3-methylphenyl)ethan-1-one
methyl 2-{1-[(2,3,5-trifluorophenyl)carbamoyl]pyrrolidin-3-yl}acetate
methyl 3-(furan-2-amido)-5-{[(2-methyl-1H-imidazol-4-yl)methyl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-6-[1-(4-methylphenyl)cyclopropanecarbonyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-phenyl-2-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]morpholine
1-(4-chloro-2-fluorobenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{1-[(4-fluorophenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
6-[(2,5-dimethylphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-(propan-2-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidin-2-amine
N-cyclooctyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
(1S,5R)-6-(4-methyl-1,3-thiazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-acetylthiophen-3-yl)-N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]acetamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-(1H-pyrazol-1-yl)propan-2-yl]amine
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyridin-2-amine
2-(1-propylpiperidin-4-yl)-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]ethan-1-one
(3-benzyl-1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl)methanol
N-{[4-hydroxy-1-(1H-pyrazole-3-carbonyl)azepan-4-yl]methyl}benzenesulfonamide
1,4-dimethyl 2-[({2-[(2-chlorophenyl)methoxy]-7-(methylsulfanyl)quinolin-3-yl}methyl)amino]butanedioate
2-amino-1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
7-(cyclobutylmethyl)-2-(2-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-8-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclohexyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
9-[2-(ethylsulfanyl)propanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
dimethyl[(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-oxazepan-6-yl)methyl]amine
1-(1-methyl-1H-pyrazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
methyl 4-[(5-{[2-(adamantan-1-yl)ethyl](methyl)amino}-2-oxoazepan-1-yl)methyl]benzoate
6-methyl-2-(4-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-hydroxycyclohexane-1-carboxamide
methyl 3-(2-methoxyacetamido)-1-(3-methylbutyl)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(pyridin-2-ylmethyl)piperazine
N-(2-methoxypyridin-3-yl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-2-carboxamide
1-(3-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
6-methyl-2-[2-({1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}amino)ethyl]-3,4-dihydropyrimidin-4-one
2-{1-[(2-ethoxyphenyl)methyl]-4-(quinolin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
3,6-dimethyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1-benzofuran-2-carboxamide
1-[(2,5-dimethoxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-chloro-4-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
1-[5-(5-fluoro-2-methoxyphenyl)furan-2-carbonyl]pyrrolidine
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(4-methoxy-3-methylphenyl)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
2-{3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-N-methylacetamide
2-{3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
N,N-dimethyl-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}azepan-4-amine
methyl 3-(pyrazine-2-amido)-5-[2-(trifluoromethyl)benzenesulfonamidomethyl]benzoate
N-[(1-{[4-(benzyloxy)phenyl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
1-(2,2-dimethylpropyl)-4-({2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)pyrrolidin-2-one
4-[4-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)piperazin-1-yl]phenol