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4-[4-({[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]-2-methylbut-3-yn-2-ol
3-phenyl-N-{1-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
3-(4-fluorophenyl)-3-{[3-(1H-pyrazol-1-yl)phenyl]formamido}propanoic acid
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
4-[(3-aminopropyl)sulfamoyl]-N-(1H-imidazol-2-ylmethyl)-N-methylbenzamide
1-methanesulfonyl-4-(3-methoxypropanoyl)-1,4-diazepane-6-carboxylic acid
5-(2,3-dimethylquinoxaline-6-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
10-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-ethyl-N-methylpyrimidine-5-carboxamide
1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxylic acid
[2-ethoxy-5-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]methyl acetate
1-{4-methoxy-2-[3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-pyrazole
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-(thiomorpholin-4-yl)propan-1-one
4-[2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)acetyl]-1-phenylpiperazin-2-one
3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-[3-(oxolan-3-yl)propyl]urea
N,N-diethyl-4-{[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}aniline
3-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-(1-{6-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
4-ethyl-3-{1-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidine
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-1-methylazepane-2-carboxamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indazol-3-yl)acetamide
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N,N,5,6-tetramethylpyrimidin-2-amine
methyl 3-[3-(dimethylamino)benzoyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(3,3-diphenylpropyl)-6-[2-(2-fluorophenyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
N-benzyl-6-[3-(methoxymethyl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[(1-cycloheptylpiperidin-3-yl)sulfamoyl]-N-methylbenzamide
8-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-{[3-cyclopropyl-1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-(2,8-dimethylquinoline-4-carbonyl)-3,9-diazaspiro[5.5]undecane
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2-(4-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]ethan-1-one
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-(4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazin-1-yl)phenol
1-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-3-ol
2-amino-4-[(3,3-dimethylbutyl)amino]quinazoline-6-carboxylic acid
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(2-fluorophenyl)-1-methylpyrrolidine-3-carboxamide
(1R,9S)-5-amino-12-methyl-3-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
5-fluoro-2-(2-{1-methyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)-1H-1,3-benzodiazole
8-[2-(3-chloro-4-hydroxyphenyl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
6-amino-N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]pyridine-3-carboxamide
4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]pyridin-2-amine
6-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-propylpyrimidin-4-amine
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
N4-[(2,3-difluoro-4-methoxyphenyl)methyl]-5-methylpyrimidine-2,4-diamine
(2S,4R)-4-amino-1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-N-methylpyrrolidine-2-carboxamide
(1R,3s,6r,8S)-4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
N-cyclopropyl-2-(4-{[(2-fluoro-4-methoxyphenyl)carbamoyl]amino}piperidin-1-yl)acetamide